Eganelisib (IPI-549): Selectivity & Specificity

Eganelisib (IPI-549) is a potent inhibitor of PIK3CG (7.9–83 nM), ABCB1. Eganelisib (IPI-549) exhibits the greatest inhibitory potency toward PIK3CG (IC50 = 7.9–83 nM).