BMS-927711 is a potent CGRP receptor antagonist. It affects cAMP signaling by blocking CGRP, to inhibit vasorelaxation.
Comprehensive IC50 Values for BMS-927711 (Rimegepant) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
BMS-927711 is a potent CGRP receptor antagonist. It affects cAMP signaling by blocking CGRP, to inhibit vasorelaxation.