BI-2865: Selectivity & Specificity
BI-2865 is a potent inhibitor of P-gp (0.3 µM), KRAS (4.3 nM). BI-2865 exhibits the greatest inhibitory potency toward KRAS (IC50 = 4.3 nM).
BI-2865 is a potent inhibitor of P-gp (0.3 µM), KRAS (4.3 nM). BI-2865 exhibits the greatest inhibitory potency toward KRAS (IC50 = 4.3 nM).