Cell-free Assays (IC50/Ki) for ARN-509 (Apalutamide)
| Key Target | IC50 (Cell-free) | Description | Reference |
|---|---|---|---|
Cell-based Assay (IC50) for ARN-509 (Apalutamide)
| Cell Type | IC50 (Cell-based) | Description | Reference |
|---|---|---|---|
| PC cells | 93 nM | Inhibition constant value for blocking AR function and testosterone-induced nuclear translocation | Download PDF |
Check the
ARN-509 (Apalutamide)
product page for in-depth specifications, including solubility, stock solutions, MOA, and working concentrations.
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- ARN-509 (Apalutamide) Mechanism of Action: Androgen Receptor Inhibition in Prostate Cancer Cell Research
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- ARN-509 (Apalutamide) Working Concentration | Cell Culture | Treatment
- ARN-509 (Apalutamide) Solubility in DMSO
- ARN-509 (Apalutamide) Stock Solution
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- ARN-509 (Apalutamide) Stability
- ARN-509 (Apalutamide) Combination Database
- ARN-509 (Apalutamide) Molecular Weight
- ARN-509 (Apalutamide) SMILES
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- ARN-509 (Apalutamide) Chemical Structure (2D and 3D)
- ARN-509 (Apalutamide) Sigma (AMBH2D6FA54D)? Try a better option.
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- ARN-509 (Apalutamide) SDS|MSDS