4-Hydroxytamoxifen is a potent, selective ER antagonist. It blocks ER signaling by binding ER, inhibiting tumor growth.
Comprehensive IC50 Values for 4-Hydroxytamoxifen (Afimoxifene) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
4-Hydroxytamoxifen is a potent, selective ER antagonist. It blocks ER signaling by binding ER, inhibiting tumor growth.