PKG inhibitor peptide is an ATP-competitive inhibitor of cGMP-dependent protein kinase (PKG), with a Ki of 86 μM.

Amino-acid Sequence

CAS No. 82801-73-8

Batch: P115301 DMSO] 100 mg/mL] false] Water] 100 mg/mL] false] Ethanol] 2 mg/mL] false Purity: 99.29%

99.29

Storage (From the date of receipt)	3 years-20°C powder	Storage of Stock Solutions Aliquot the stock solutions to avoid repeated freeze-thaw cycles	1 year-80°Cin solvent
			1 month-20°Cin solvent

In vitro
Batch:

DMSO : 100 mg/mL ( (106.03 mM)； Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Water : 100 mg/mL

Ethanol : 2 mg/mL

In vivo
Batch:

Add solvents to the product individually and in order.

Description

PKG inhibitor peptide is an ATP-competitive inhibitor of cGMP-dependent protein kinase (PKG), with a Ki of 86 μM.

Targets

PKG

86 μM

References
[1] Bhatnagar D, et al. Biochemistry. 1988 Mar 22;27(6):1988-94.

References

Molecular Formula:	C₃₈H₇₄N₁₈O₁₀
Molecular Weight:	943.11
CAS No.:	82801-73-8
Appearance:	White Powder
Peptide Content (by %N):	≥80%
Single Impurity (by HPLC):	≤1.0%
Assay (By Anhydrous, Acetic Acid-free):	95.0~105.0%
MS:	Consistent
Packing:	plastic vial(dedicated for peptide packing) or glass vial, quantity according to customer's detail requirement.
Storage (From the date of receipt):	3 years-20°C powder
Shipping:	Room temperature shipping(Stability testing shows this product can be shipped without any cooling measures.)