G9a/GLP Inhibitors

Cat.No. Product Name Information Product Use Citations Product Validations
S7020 UNC0646 UNC0646 is a selective histone lysine methyltransferase (HMTase) inhibitor for G9a and GLP with IC50 of 6 nM and 15 nM , respectively, with excellent potency in a variety of cell lines and excellent separation of functional potency versus cell toxicity.
PhD Thesis, Universiteit van Amsterdam, 2025, 83-85
Journal of Orthopaedic Translation, 2024, 211-225
Genome Instability & Disease, 2022, 21