Home Metabolism -Proteases SGK SGK1 Selective Inhibitors

SGK1 Selective Inhibitors

  • SGK1
  • SGK2
  • SGK3
Catalog No. Product Name Information Selective / Pan IC50 / Ki
S8824 EMD638683 EMD638683 is a highly selective inhibitor of serum- and glucocorticoid-inducible kinase 1 (SGK1) with IC50 of 3 μM. EMD638683 exhibits antihypertensive potency and anti-tumor activity. Selective SGK1, IC50: 3 μM
S7209 GSK650394 GSK650394 is a serum- and glucocorticoid-regulated kinase-1 inhibitor with IC50 of 62 nM and 103 nM for SGK1 and SGK2, respectively. Pan SGK1, IC50: 62 nM