Home Metabolism PDE PDE10A Selective Inhibitors

PDE10A Selective Inhibitors

  • PDE1
  • PDE2
  • PDE3
  • PDE4
  • PDE5
  • PDE6
  • PDE10A
  • PDE9
  • PDE4B
Catalog No. Product Name Information Selective / Pan IC50 / Ki
S8459 TAK-063 TAK-063 (Balipodect) is a novel and selective phosphodiesterase 10A(PDE10A) inhibitor with an IC50 of 0.30 nM. Selective PDE10A, IC50: 0.3 nM
S2687 Mardepodect (PF-2545920) Mardepodect (PF-2545920) is a potent and selective PDE10A inhibitor with IC50 of 0.37 nM, with >1000-fold selectivity over the PDE. Selective PDE10A, IC50: 0.37 nM