Home Metabolism -Cell Cycle Serine/threonin kinase GAK Selective Inhibitors

GAK Selective Inhibitors

  • serine/threonine kinase
  • STK
  • WNK
  • DCLK
  • GCN
  • GAK
  • SRPK
  • PASK
  • BUB1
Catalog No. Product Name Information Selective / Pan IC50 / Ki
S6710 SGC-GAK-1 SGC-GAK-1 is a potent, selective, and cell-active inhibitor of cyclin G-associated kinase (GAK) with Ki value of 3.1 nM and >50-fold selectivity over nearest kinase. Selective GAK, Ki: 3.1 nM
S0848 GAK inhibitor 49 GAK inhibitor 49 is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with an IC50 of 56 nM. Selective GAK, IC50: 56 nM