Home GPCR & G Protein cAMP EPAC1 Inhibitors | Antagonists

EPAC1 Inhibitors | Antagonists

  • AC
  • EPAC1
  • EPAC2
  • PACAP receptor
Catalog No. Product Name Information Selective / Pan IC50 / Ki
S0837 HJC0197 HJC0197 is a selective Epac 1/2 dual antagonists with an IC50 of 5.9 μM for Epac2. Pan
S7499 ESI-09 ESI-09 is a specific exchange protein directly activated by cAMP (EPAC) inhibitor with IC50 of 3.2 μM and 1.4 μM for EPAC1 and EPAC2, respectively, >100-fold selectivity over PKA. Pan EPAC1, IC50: 3.2 μM