Home Metabolism CPT CPT1 Selective Inhibitors

CPT1 Selective Inhibitors

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S6959 Perhexiline maleate Perhexiline maleate is a potent inhibitor of carnitine palmitoyltransferase 1 (CPT1) with IC50s of 77 μM and 148 μM for rat heart CPT1 and liver CPT1, respectively, and also inhibits carnitine palmitoyltransferase 2 (CPT2). Selective rat heart CPT1, IC50: 77 μM; rat liver CPT1, IC50: 148 μM