Home Metabolism -Cell Cycle Serine/threonin kinase BUB1 Selective Inhibitors

BUB1 Selective Inhibitors

  • serine/threonine kinase
  • STK
  • WNK
  • DCLK
  • GCN
  • GAK
  • SRPK
  • PASK
  • BUB1
Catalog No. Product Name Information Selective / Pan IC50 / Ki
S3522 2OH-BNPP1 2OH-BNPP1 is an inhibitor of the kinase activity of BUB1 (budding uninhibited by benzimidazoles-1, BUB1 Mitotic Checkpoint Serine/Threonine Kinase) that can be used for the treatment of cancer. Selective
S8945 BAY-1816032 BAY-1816032 is a potent and oral available inhibitor of budding uninhibited by benzimidazoles 1 (BUB1) kinase with IC50 of 6.1 nM for recombinant catalytic domain of human BUB1. BAY-1816032 has antitumor activity. Selective BUB1, IC50: 6.1 nM