AKR1C3 Inhibitors

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S0764 AKR1C1-IN-1

AKR1C1-IN-1 is a potent and selective inhibitor of human 20alpha-hydroxysteroid dehydrogenase (AKR1C1) with Ki of 4 nM, 87 nM, 4.2 μM and 18.2 μM for AKR1C1, AKR1C2, AKR1C3 and AKR1C4, respectively.

Pan AKR1C3, Ki: 4.2 μM