Target Selectivity of Vactosertib (TEW-7197)

Key TargetIC50DescriptionReference
TGF-β RI/ALK-5 12.9 nM Kinase activity assay PMC8022551
ALK5 12.9 nM kinase activity inhibition PMC8158184
ALK-2 17.3 nM Kinase activity assay PMC8022551
ALK-4 17.3 nM Kinase activity assay PMC8022551
ALK2 17.3 nM kinase activity inhibition PMC8158184
Check the Vactosertib (TEW-7197) product page for in-depth specifications, including solubility, stock solutions, MOA, and working concentrations.

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