AMD3100 (Plerixafor): Selectivity & Specificity

AMD3100 (Plerixafor) is a potent inhibitor of Escherichia coli S30 extract system (62.30 ±6.47mM), CXCR4 (11.4 µM), TGFβ-1 (9.1 µM). AMD3100 (Plerixafor) exhibits the greatest inhibitory potency toward TGFβ-1 (IC50 = 9100 nM).