Pexidartinib is an ATP-competitive CSF-1R inhibitor. It blocks PI3K/AKT signaling by preventing ATP entry, halting tumor growth.
Comprehensive IC50 Values for Pexidartinib (PLX3397) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Pexidartinib is an ATP-competitive CSF-1R inhibitor. It blocks PI3K/AKT signaling by preventing ATP entry, halting tumor growth.