JPH203 (Nanvuranlat) is a selective, competitive LAT1 inhibitor. It affects mTORC1 and ATF4/CHOP signaling pathways by blocking LAT1-mediated essential amino acid uptake, effectively inhibiting cancer cell proliferation, viability, and migration.
Comprehensive IC50 Values for JPH203 (Nanvuranlat) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
JPH203 (Nanvuranlat) is a selective, competitive LAT1 inhibitor. It affects mTORC1 and ATF4/CHOP signaling pathways by blocking LAT1-mediated essential amino acid uptake, effectively inhibiting cancer cell proliferation, viability, and migration.