|
SU-DIPG-36
|
15.87 µM
|
Crystal violet (CV) assay
|
Download PDF
|
|
HGC-27
|
3.35 ± 0.15 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
AGS
|
> 10.00 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
FU97
|
0.48 ± 0.27 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
MKN1
|
0.15 ± 0.06 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
MKN1
|
3.98 ± 0.67 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
MKN74
|
1.22 ± 0.22 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
MKN74
|
8.39 ± 0.04 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
NCI-N87
|
0.004 ± 0.001 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
NCI-N87
|
0.013 ± 0.001 µM
|
Sulforhodamine B (SRB) colorimetric assay; non-linear least squares curve fitting (four-parameter analysis, log (inhibitor) vs. response, variable slope) using Gen5 software ([Vendor], UK).
|
PMC10965263
|
|
OE19
|
> 1 μM
|
Crystal violet staining
|
Download PDF
|
|
4NQO-L cells
|
0.021 μM
|
crystal violet staining, absorbance measured at 570 nm
|
Download PDF
|
|
LN-18
|
1.08 µM
|
SRB colorimetric assay, non-linear least squares curve fitting
|
PMC11092418
|
|
A172
|
10.00 µM
|
SRB colorimetric assay, non-linear least squares curve fitting
|
PMC11092418
|
|
U118MG
|
5.60 µM
|
SRB colorimetric assay, non-linear least squares curve fitting
|
PMC11092418
|
|
T-98G
|
3.25 µM
|
SRB colorimetric assay, non-linear least squares curve fitting
|
PMC11092418
|
|
LN-18
|
8.55 µM
|
SRB colorimetric assay, non-linear least squares curve fitting
|
PMC11092418
|
|
A172
|
10.00 µM
|
SRB colorimetric assay, non-linear least squares curve fitting
|
PMC11092418
|
|
U118MG
|
6.39 µM
|
SRB colorimetric assay, non-linear least squares curve fitting
|
PMC11092418
|
|
T-98G
|
10.00 µM
|
SRB colorimetric assay, non-linear least squares curve fitting
|
PMC11092418
|
|
Jurkat Cells
|
1.43 ±0.35µM
|
MTT assay
|
Download PDF
|
|
PBMCs
|
12.71 ±2.08µM
|
MTT assay
|
Download PDF
|
|
HCC1954
|
2.42 ± 0.30 μM
|
MTT assay, nonlinear regression modeling via GraphPad Prism software
|
Download PDF
|
|
hFB-hTERT
|
12.80 ± 1.41 μM
|
MTT assay, nonlinear regression modeling via GraphPad Prism software
|
Download PDF
|
|
TT cells
|
1.2 ×10−9 M
|
real-time cell analysis system (xCELLigence System) and nonlinear regression analysis (Sigmoidal dose–response [variable slope])
|
Download PDF
|
|
muPC
|
4.61 µM
|
Cell Counting Kit-8 and MTT assays, viability determined by absorbance at 450 nm, IC50 calculated using a specific formula.
|
PMC11199751
|
|
bePC
|
7.47 µM
|
Cell Counting Kit-8 and MTT assays, viability determined by absorbance at 450 nm, IC50 calculated using a specific formula.
|
PMC11199751
|
|
MCF-7
|
~17µM
|
MTT assay, nonlinear regression (curve fit) in log inhibitor vs response-variable slope (four parameters) equation.
|
PMC12118019
|
|
SK-BR-3
|
77 nM
|
dose-response studies
|
Download PDF
|
|
SK-BR-3
|
150 nM
|
Sulforhodamine B (SRB) colorimetric assay
|
Download PDF
|
|
SK-BR-3_LR600
|
600 nM
|
Sulforhodamine B (SRB) colorimetric assay
|
Download PDF
|
|
A549
|
11.57 µM
|
MTT assay
|
Download PDF
|
|
SKOV-3
|
16.95 µM
|
MTT assay
|
Download PDF
|
|
SK-BR-3
|
8.54 µM
|
MTT assay
|
Download PDF
|
|
MRC-5
|
43.94 µM
|
MTT assay
|
Download PDF
|
|
SKBR3-LR
|
212 nmol/L
|
Cell growth assay (DAPI staining and nuclei counting)
|
PMC11145169
|
|
GDSC cell lines (for THCA patients)
|
Lower IC50 values in patients with high LNM potential and hi
|
oncoPredict algorithm (Ridge regression) based on GDSC database
|
Download PDF
|
|
SK-BR3
|
800 nM
|
MTT assay
|
Download PDF
|
|
SK-BR3
|
500 nM
|
MTT assay
|
Download PDF
|
|
SK-BR3
|
100 nM
|
MTT assay
|
Download PDF
|
|
SK-BR-3
|
0.001 µM
|
MTT cell proliferation assay
|
Download PDF
|
|
T47D
|
0.001 µM
|
MTT cell proliferation assay
|
Download PDF
|
|
Hs578T
|
10 µM
|
MTT cell proliferation assay
|
Download PDF
|
|
ZR75
|
0.001 µM
|
MTT cell proliferation assay
|
Download PDF
|
|
BT549
|
10 µM
|
MTT cell proliferation assay
|
Download PDF
|
|
MDA-MB-231
|
10 µM
|
MTT cell proliferation assay
|
Download PDF
|
|
MDA-MB-468
|
10 µM
|
MTT cell proliferation assay
|
Download PDF
|
|
MX-1
|
10 µM
|
MTT cell proliferation assay
|
Download PDF
|
|
HROP68Tu2 cells
|
6.27 μM
|
Crystal violet assay
|
Download PDF
|
|
SH-SY5Y
|
36.9 µM
|
MTT assay, CalcuSyn software
|
Download PDF
|
|
SH-SY5Y
|
9.7 µM
|
MTT assay, CalcuSyn software
|
Download PDF
|
|
SK-N-BE(2)
|
27.2 µM
|
MTT assay, CalcuSyn software
|
Download PDF
|
|
SK-N-BE(2)
|
8.3 µM
|
MTT assay, CalcuSyn software
|
Download PDF
|
|
DAOY
|
10.0 µM
|
MTT assay, CalcuSyn software
|
Download PDF
|
|
Saos-2
|
11.9 µM
|
MTT assay, CalcuSyn software
|
Download PDF
|
|
RD
|
8.7 µM
|
MTT assay, CalcuSyn software
|
Download PDF
|
|
BT474 (TSC2-NC)
|
0.2583 μM
|
Cell Counting Kit 8 (CCK8)
|
Download PDF
|
|
BT474 (TSC2-WT)
|
0.2919 μM
|
Cell Counting Kit 8 (CCK8)
|
Download PDF
|
|
BT474 (TSC2-MT)
|
1.416 μM
|
Cell Counting Kit 8 (CCK8)
|
Download PDF
|
|
CTOS
|
1.8 μM
|
ATP content measured with Luminescent Cell Viability Assays
|
Download PDF
|
|
UM-SCC-11B
|
8.843 µM
|
Alamar Blue viability assay; Graph Pad Prism
|
PMC9021830
|
|
UM-SCC-22B
|
8.433 µM
|
Alamar Blue viability assay; Graph Pad Prism
|
PMC9021830
|
|
PfNF54
|
0.26 ± 0.07 µM
|
Plasmodium Lactate Dehydrogenase (pLDH) Assay.
|
Download PDF
|
|
PfK1
|
0.85 ± 0.02 µM
|
Plasmodium Lactate Dehydrogenase (pLDH) Assay.
|
Download PDF
|
|
Vero cells
|
31.1 µM
|
SARS-CoV-2 reporter virus (mNeon) infection assay
|
Download PDF
|
|
SUN216 cells
|
0.24 nM
|
CCK-8 assay
|
PMC8799157
|
|
SUN216/LR cells
|
>10 nM
|
CCK-8 assay
|
PMC8799157
|
|
SK-BR-3
|
1.12 × 10−12 M
|
AlamarBlue cell viability reagent
|
Download PDF
|
|
SKBR3-HO-1
|
4.31 × 10−8 M
|
AlamarBlue cell viability reagent
|
Download PDF
|
|
NCI-N87
|
39.8 ± 13.3 nM
|
acid phosphatase assay
|
Download PDF
|
|
ESO26
|
290.8 ± 42.7 nM
|
acid phosphatase assay
|
Download PDF
|
|
OE19
|
1660 ± 151.7 nM
|
acid phosphatase assay
|
Download PDF
|
|
SNU16
|
> 10,000 nM
|
MTS assay
|
Download PDF
|
|
KATOIII
|
> 10,000 nM
|
acid phosphatase assay
|
Download PDF
|
|
HT-29
|
6.81±1.24 μM
|
Sulforhodamine B (SRB) assay
|
PMC6717862
|
|
HCC-1954
|
2.3 ± 0.2 mM
|
MTT assay
|
Download PDF
|
|
MCF-10A
|
4.6 ± 0.2 mM
|
MTT assay
|
Download PDF
|
|
SKOV3 SYK130E Tet-off cells (SYK130E induced)
|
150.8 μM
|
CellTiter-Glo® 3D Cell Viability Assay
|
PMC6796592
|
|
81-II
|
321 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
H-ICN
|
3188 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
2-59LR
|
11271 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
84WS
|
799 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
6-CEH
|
1026 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
B2C-UNS
|
5938 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
7365
|
222 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
28J
|
75181 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
HEC-1
|
31600 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
HEC-1-B
|
31600 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
152-CEH
|
3701 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
DLD-1
|
14634 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
uDaF
|
542 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
HCT-15
|
11829 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
3-CU-MU
|
613 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
PMA 565-UA
|
492 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
PMA 3-RB-KS
|
251 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
PMA 474-TB
|
262 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
PMA 4591CCH
|
6241 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
PMA 883A
|
1021 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
PMA 02-TB
|
80251 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
PMA 864-BM-ADM
|
1 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
AU-565
|
125 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
BT-474
|
3062 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
HCC1954
|
294 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
MDA-MB-453
|
2844 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
SK-BR-3
|
152 nM
|
Cell proliferation assays measured by ATPlite 1Step luminescence, calculated by non-linear regression using IDBS XLfit 5.
|
Download PDF
|
|
Caski
|
0.54 ± 0.023 µM
|
Cell Titer96 Aqueous cell proliferation assay, nonlinear regression analysis using GraphPad Prism software
|
PMC5327645
|
|
C-33A
|
1.78 ± 0.43 µM
|
Cell Titer96 Aqueous cell proliferation assay, nonlinear regression analysis using GraphPad Prism software
|
PMC5327645
|
|
SiHa
|
2.36 ± 0.63 µM
|
Cell Titer96 Aqueous cell proliferation assay, nonlinear regression analysis using GraphPad Prism software
|
PMC5327645
|
|
HeLa
|
2.19 ± 0.98 µM
|
Cell Titer96 Aqueous cell proliferation assay, nonlinear regression analysis using GraphPad Prism software
|
PMC5327645
|
|
ZR-75-30
|
50-100 nM
|
CellTiter 96 Aqueous Non-Radioactive Cell Proliferation Assay (MTS)
|
Download PDF
|
|
BT474
|
50-100 nM
|
CellTiter 96 Aqueous Non-Radioactive Cell Proliferation Assay (MTS)
|
Download PDF
|
|
AU-565
|
50-100 nM
|
CellTiter 96 Aqueous Non-Radioactive Cell Proliferation Assay (MTS)
|
Download PDF
|
|
MDA-MB-361
|
~1 μM
|
CellTiter 96 Aqueous Non-Radioactive Cell Proliferation Assay (MTS)
|
Download PDF
|
|
MDA-MB-453
|
10 μM
|
CellTiter 96 Aqueous Non-Radioactive Cell Proliferation Assay (MTS)
|
Download PDF
|
|
HCC1806
|
100 nM
|
Growth inhibition (SRB assay), Annexin-V apoptotic signal
|
Download PDF
|
|
LIM1215-HER2
|
>10 μM
|
clonogenic assay
|
Download PDF
|
|
SW48-HER2
|
>10 μM
|
clonogenic assay
|
Download PDF
|
|
PC12 cells (EGFR)
|
305 nM
|
Split TEV recruitment assay, luciferase activity
|
Download PDF
|
|
A549 cells (EGFR)
|
21.87 nM
|
Western blotting, p-EGFR-Y1068 antibody
|
Download PDF
|
|
T-47D cells (ERBB4)
|
53.70 nM
|
Western blotting, p-ERBB4-Y1284 antibody
|
Download PDF
|
|
BT-474
|
0.0178 ± 0.00285 μM
|
CellTiter 961AQueous One Solution Cell Proliferation Assay (MTS assay)
|
Download PDF
|
|
BT-474-R
|
0.239 ± 0.0443 μM
|
CellTiter 961AQueous One Solution Cell Proliferation Assay (MTS assay)
|
Download PDF
|
|
JIMT-1 cells
|
~1.5 µM
|
Viability assay (crystal violet staining, absorbance 540 read)
|
Download PDF
|
|
SK-BR-3
|
120 nM
|
MTT assay
|
Download PDF
|
|
SK-BR-3
|
120 nM
|
MTT assay
|
Download PDF
|
|
SK-BR-3
|
120 nM
|
MTT assay
|
Download PDF
|
|
SK-BR-3
|
120 nM
|
MTT assay
|
Download PDF
|
|
SK-BR-3
|
120 nM
|
MTT assay
|
Download PDF
|
|
SK-BR-3
|
120 nM
|
MTT assay
|
Download PDF
|
|
SK-BR-3
|
120 nM
|
MTT assay
|
Download PDF
|
|
SKBR3-L
|
6.5 ± 0.4 μM
|
Proliferation assay
|
Download PDF
|
|
HCC1954-L
|
2.67 ± 0.08 μM
|
Proliferation assay
|
Download PDF
|
|
MCF7mock
|
40 μM (24h), 19.6 μM (48h)
|
MTT assay
|
Download PDF
|
|
MCF7G6PD+
|
51 μM (24h), 37.6 μM (48h)
|
MTT assay
|
Download PDF
|
|
NZBR1
|
>1000 nM
|
thymidine incorporation assay
|
Download PDF
|
|
NZBR2
|
>1000 nM
|
thymidine incorporation assay
|
Download PDF
|
|
NZBR3
|
1.2 nM
|
thymidine incorporation assay
|
Download PDF
|
|
NZBR4
|
>1000 nM
|
thymidine incorporation assay
|
Download PDF
|
|
SK-BR-3
|
1.5 nM
|
thymidine incorporation assay
|
Download PDF
|
|
MDA-MB-231
|
>1000 nM
|
thymidine incorporation assay
|
Download PDF
|
|
ZR75.1
|
>1000 nM
|
thymidine incorporation assay
|
Download PDF
|
|
HCC1954-Par
|
273 nM
|
acid phosphatase assay
|
PMC5344284
|
|
HCC1954-NR
|
2.7 mM
|
acid phosphatase assay
|
PMC5344284
|
|
EFM192A-Par
|
50 nM
|
acid phosphatase assay
|
PMC5344284
|
|
EFM192A-NR
|
7.97 mM
|
acid phosphatase assay
|
PMC5344284
|
|
HCC1569 (PIK3CA WT) ERBB4-WT
|
514.02 nM
|
Proliferation assays over 5 days
|
PMC6047239
|
|
HCC1569 (PIK3CA WT) ERBB4-V721I
|
503.67 nM
|
Proliferation assays over 5 days
|
PMC6047239
|
|
HCC1569 (PIK3CA WT) ERBB4-S303F
|
736.41 nM
|
Proliferation assays over 5 days
|
PMC6047239
|
|
BT474 (PIK3CA mutated) ERBB4-WT
|
42.69 nM
|
Proliferation assays over 5 days
|
PMC6047239
|
|
BT474 (PIK3CA mutated) ERBB4-V721I
|
44.78 nM
|
Proliferation assays over 5 days
|
PMC6047239
|
|
HCC1954 (PIK3CA mutated) ERBB4-WT
|
894.24 nM
|
Proliferation assays over 5 days
|
PMC6047239
|
|
HCC1954 (PIK3CA mutated) ERBB4-V721I
|
789.48 nM
|
Proliferation assays over 5 days
|
PMC6047239
|
|
SK-BR-3
|
1.444 μM
|
formazan dye assay, sigmoidal curves calculated with Boltzmann equation
|
Download PDF
|
|
T47D
|
9.082 μM
|
formazan dye assay, sigmoidal curves calculated with Boltzmann equation
|
Download PDF
|
|
Jurkat
|
20.091 μM
|
formazan dye assay, sigmoidal curves calculated with Boltzmann equation
|
Download PDF
|
|
CNE-2
|
3–5 μM
|
Cell Counting Kit-8 (CCK-8) assay
|
PMC5067011
|
|
HONE-1
|
3–5 μM
|
Cell Counting Kit-8 (CCK-8) assay
|
PMC5067011
|
|
HCC38
|
9.2 μM
|
MTT cell viability assay
|
Download PDF
|
|
MCF7/BCAR4
|
7–9 mM
|
WST-1 proliferation assays, estimated by sigmoid inhibitory effect models 107 and 108 as implemented in the software programme Phoenix WinNonLin 6.1.
|
PMC3464772
|
|
MCF7/vector
|
8–12 mM
|
WST-1 proliferation assays, estimated by sigmoid inhibitory effect models 107 and 108 as implemented in the software programme Phoenix WinNonLin 6.1.
|
PMC3464772
|
|
SK-BR-3
|
<0.1mM
|
Not explicitly stated, inferred from sensitivity description
|
PMC5680796
|
|
JIMT1 parental cells
|
7.0±1.0 µmol/L
|
MTT-based cell viability assays
|
Download PDF
|
|
control-shRNA/JIMT1 cells
|
7.5±1.0 µmol/L
|
MTT-based cell viability assays
|
Download PDF
|
|
ATG12-shRNA/JIMT1 cells
|
0.7±0.4 µmol/L
|
MTT-based cell viability assays
|
Download PDF
|
|
786-O
|
4.6 μM
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MTT proliferation assays
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Download PDF
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HT-29
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2.1 μM
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MTT proliferation assays
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Download PDF
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HT-29 SUN
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4.2 μM
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MTT proliferation assays
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Download PDF
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SKBR3-P
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57.3 ± 6.6 nM
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Proliferation measured using the acid phosphatase assay, IC50 calculated using CalcuSyn software.
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Download PDF
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SKBR3-L
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1237.7 ± 212.7 nM
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Proliferation measured using the acid phosphatase assay, IC50 calculated using CalcuSyn software.
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Download PDF
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SKBR3-T
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79.3 ± 12.5 nM
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Proliferation measured using the acid phosphatase assay, IC50 calculated using CalcuSyn software.
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Download PDF
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HCC1954-P
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581.0 ± 84.5 nM
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Proliferation measured using the acid phosphatase assay, IC50 calculated using CalcuSyn software.
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Download PDF
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HCC1954-L
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3602.0 ± 311.3 nM
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Proliferation measured using the acid phosphatase assay, IC50 calculated using CalcuSyn software.
|
Download PDF
|
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BT474-P
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14.3 ± 5.0 nM
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Proliferation measured using the acid phosphatase assay, IC50 calculated using CalcuSyn software.
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Download PDF
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BT474-RES
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223.7 ± 48.5 nM
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Proliferation measured using the acid phosphatase assay, IC50 calculated using CalcuSyn software.
|
Download PDF
|
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UM-SCC-47
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0.36 µM
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The viable cell number was determined using a 10% concentration of UptiBlue reagent ([Vendor], France). The analyses were performed by fluorimetry and normalized to a non-treated control.
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PMC4322874
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SCC-154
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0.02 µM
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The viable cell number was determined using a 10% concentration of UptiBlue reagent ([Vendor], France). The analyses were performed by fluorimetry and normalized to a non-treated control.
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PMC4322874
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BT474
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0.036 ± 0.0151 μM
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Acid Phosphatase assay
|
Download PDF
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SK-BR-3
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0.080 ± 0.0173 μM
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Acid Phosphatase assay
|
Download PDF
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EFM192A
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0.193 ± 0.0665 μM
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Acid Phosphatase assay
|
Download PDF
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HCC1954
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0.4166 ± 0.18 μM
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Acid Phosphatase assay
|
Download PDF
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MDAMB453
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6.08 ± 0.825 μM
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Acid Phosphatase assay
|
Download PDF
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MDAMB231
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7.46 ± 0.102 μM
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Acid Phosphatase assay
|
Download PDF
|
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BT474 (pHER2)
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0.0411 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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BT474 LR (pHER2)
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0.0204 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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BT474 wt (pHER2)
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0.0798 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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BT474 E545K (pHER2)
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0.0852 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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BT474 H1047R (pHER2)
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0.0978 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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SKBR3 (pHER2)
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0.0254 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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SKBR3 wt (pHER2)
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0.0297 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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SKBR3 E545K (pHER2)
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0.0211 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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SKBR3 H1047R (pHER2)
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0.0241 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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MDA361 (pHER2)
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0.0160 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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HCC1954 (pHER2)
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0.0681 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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SUM190 (pHER2)
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0.0465 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
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UACC893 (pHER2)
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0.0444 μM
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PathScan Sandwich ELISA for pHER2, followed by log(inhibitor) vs. response curves using a variable slope model and GraphPad Prism software.
|
Download PDF
|
