Target Selectivity of GSK2606414
| Key Target | IC50 | Description | Reference |
|---|---|---|---|
| RIPK1 | 1 µM | Off-target activity | PMC12838581 |
| c-kit | 1 µM | Off-target activity | PMC12838581 |
| AuroraBkinase | 1 µM | Off-target activity | PMC12838581 |
| BRK | 1 µM | Off-target activity | PMC12838581 |
| MAP3K10 | 1 µM | Off-target activity | PMC12838581 |
| c-MER | 1 µM | Off-target activity | PMC12838581 |
| DDR2 | 1 µM | Off-target activity | PMC12838581 |
| MYLK2 | 1 µM | Off-target activity | PMC12838581 |
| IKBKE | 1 µM | Off-target activity | PMC12838581 |
| TRKC | 1 µM | Off-target activity | PMC12838581 |
| MAP3K11 | 1 µM | Off-target activity | PMC12838581 |
| RET | 1 µM | Off-target activity | PMC12838581 |
| LCK | 1 µM | Off-target activity | PMC12838581 |
| NEK4 | 1 µM | Off-target activity | PMC12838581 |
| MAP4K5 | 1 µM | Off-target activity | PMC12838581 |
| MAP3K9 | 1 µM | Off-target activity | PMC12838581 |
| TRKA | 1 µM | Off-target activity | PMC12838581 |
| AXL | 1 µM | Off-target activity | PMC12838581 |
| TRKB | 1 µM | Off-target activity | PMC12838581 |
| YES1 | 1 µM | Off-target activity | PMC12838581 |
| WNK2 | 1 µM | Off-target activity | PMC12838581 |
Check the
GSK2606414
product page for in-depth specifications, including solubility, stock solutions, MOA, and working concentrations.
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- GSK2606414 Mechanism of Action: PERK Inhibition in Neuronal Cells Research
- GSK2606414 Working Concentration | Cell Culture | Treatment
- GSK2606414 Solubility in DMSO
- GSK2606414 Stock Solution
- GSK2606414 Storage
- GSK2606414 Stability
- GSK2606414 Combination Database
- GSK2606414 Molecular Weight
- GSK2606414 SMILES
- GSK2606414 CAS Number
- GSK2606414 Chemical Structure (2D and 3D)
- GSK2606414 MedChemExpress (HY-18072)? Try a better option.
- GSK2606414 Sigma (508340)? Try a better option.
- GSK2606414 Cayman (17376)? Try a better option.
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- GSK2606414 SDS|MSDS