FK866 (Daporinad): Mechanism of Action

FK866 (Daporinad) MOA:Targeting NAMPT/NAD+ Salvage Pathway for Cancer Biology

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FK866 (Daporinad) is a potent and specific NAMPT inhibitor. It affects NAD+ biosynthesis and NF-κB signaling pathways by depleting intracellular NAD+ and ATP levels, effectively inhibiting cancer cell proliferation and promoting apoptosis.

Primary Applications and Mechanism of Action