Exarafenib (KIN-2787) is a potent, selective pan-RAF inhibitor. It affects MAPK signaling by binding RAF, inhibiting pERK.
Comprehensive IC50 Values for Exarafenib (KIN-2787) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Exarafenib (KIN-2787) is a potent, selective pan-RAF inhibitor. It affects MAPK signaling by binding RAF, inhibiting pERK.