Dasatinib is a potent ATP-competitive BCR-ABL/SRC inhibitor. It blocks MAPK signaling by binding ATP sites, inducing apoptosis.
Comprehensive IC50 Values for Dasatinib (BMS-354825) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Dasatinib is a potent ATP-competitive BCR-ABL/SRC inhibitor. It blocks MAPK signaling by binding ATP sites, inducing apoptosis.