PR-171 (Carfilzomib): Mechanism of Action

PR-171 (Carfilzomib) MOA:Targeting Proteasome/Ubiquitin-Proteasome Pathway for Multiple Myeloma Therapy

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PR-171 (Carfilzomib) is a potent, selective, and irreversible 20S proteasome inhibitor. It affects NF-κB and apoptotic signaling by binding to the β5 subunit to block polyubiquitinated protein degradation, effectively inducing apoptosis and inhibiting tumor cell proliferation.

Primary Applications and Mechanism of Action