BRM014 is a selective mutant EGFR PROTAC. It affects EGFR signaling, by CRBN-dependent degradation, to inhibit proliferation.
BRM/BRG1 ATP Inhibitor-1 (BRM014) IC50 for Cell-based and Cell-free Assays
Comprehensive IC50 Values for BRM/BRG1 ATP Inhibitor-1 (BRM014) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.