Clinical Trials

Sulfadoxine is currently being evaluated across several clinical trials investigating its utility in malaria prevention, maternal malaria during pregnancy, and bioequivalence assessments. Encompassing Phase I, Phase III, Phase IV, and unclassified trial phases, these studies are sponsored by both research networks and pharmaceutical manufacturers. Spanning recruiting, active not recruiting, and unknown recruitment statuses, these efforts underscore the ongoing clinical interest in optimizing sulfadoxine-based combination regimens for parasitic disease control.

NCT Number Recruitment Conditions Sponsor/Collaborators Start Date Phases
NCT06162078 Recruiting
Maternal Malaria During Pregnancy - Baby Not Yet Delivered
Groupe de Recherche Action en Sante|European Vaccine Initiative
2023-08-25 --
NCT05979896 Recruiting
Malaria
Malaria Consortium
2023-07-28 Phase 4
NCT05478954 Active not recruiting
Malaria
Malaria Consortium
2022-07-15 Phase 4
NCT05471544 Active not recruiting
Malaria
Malaria Consortium
2022-07-18 Phase 3
NCT04577469 Unknown status
Bioequivalence
Emzor Pharmaceutical Industries Limited
2020-12 Phase 1

(data from https://clinicaltrials.gov, updated on 2024-05-22)

Check the Sulfadoxine product page for in-depth specifications, including solubility, stock solutions, MOA, and working concentrations.

Compliance for Clinical Use

Mechanism and Biochemical Profile

Sulfadoxine competitively inhibits dihydropteroate synthase within the parasite folic acid biosynthetic pathway, thereby blocking downstream enzymatic synthesis of essential folate cofactors required for nucleic acid production. This inhibition halts intracellular replication of Plasmodium parasites, providing the mechanistic basis for its clinical utility in preventing and treating malaria and maternal malaria during pregnancy.

Appendix RUO and cGMP Quality Standards

Quality Dimension RUO (Research Use Only) cGMP (Current Good Manufacturing Practice)
Clinical Applicability Prohibited in human clinical trials or medical diagnostics. Mandatory for human clinical trials (Phase I–III) and therapies.
Regulatory Status Non-regulated grade; exempt from drug manufacturing laws. Legally enforced by health authorities (e.g., FDA, EMA, NMPA).
Facility Environment Unclassified analytical or research laboratories. Validated Cleanrooms (ISO Class 5–8) with continuous monitoring.
Quality Control Basic purity and activity testing. Rigorous safety release testing (Sterility, Endotoxin, Mycoplasma).
Process Validation Basic equipment calibration; no process validation required. Full qualification (IQ/OQ/PQ) and complete batch records.
Quality Assurance Vendor self-declared without required formal QMS. Mandatory QA/QC unit, Change Control, CAPA, and vendor audits.
Regulatory Impact High risk of IND rejection if used as a critical raw material. Required for IND/NDA filings, supported by Drug Master Files (DMF).

Footnotes

Regulatory Note: Governed by FDA (21 CFR Parts 210/211/312), EMA (EudraLex Vol 4), ICH Guidelines (E6/Q7/Q9/Q10), and compendial standards (USP <71>/<85>/<1043>).

Note: Technical data last updated: Sep 1, 2026.