Bosutinib is a potent, ATP-competitive Src/Abl kinase inhibitor. It affects BCR-ABL and Src signaling pathways by competing with ATP to inhibit kinase phosphorylation, effectively suppressing cancer cell proliferation and inducing apoptosis.
Comprehensive IC50 Values for SKI-606 (Bosutinib) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Bosutinib is a potent, ATP-competitive Src/Abl kinase inhibitor. It affects BCR-ABL and Src signaling pathways by competing with ATP to inhibit kinase phosphorylation, effectively suppressing cancer cell proliferation and inducing apoptosis.