LPA2 Antagonists

Home GPCR & G Protein LPA Receptor LPA2 Antagonists

  • LPA1
  • LPA2
  • LPA3
Catalog No. Product Name Information Selective / Pan IC50 / Ki
S1315 Ki16425 Ki16425 is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM in RH7777 cell lines, respectively, shows no activity at LPA4, LPA5, LPA6. Pan LPA2, Ki: 6.5 μM