CGRP Selective Antagonists

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S8212 Olcegepant Olcegepant (BIBN4096; BIBN4096BS) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with an IC50 of 0.03 nM. Selective CGRP, IC50: 0.03 nM