Trametinib (GSK1120212) Mechanism of Action: MEK Inhibition in Melanoma Cell Research

Trametinib (GSK1120212) MOA:Targeting MEK/MAPK for Metastatic Melanoma

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Trametinib (GSK1120212) is a highly selective, reversible allosteric MEK1/2 inhibitor. It affects the MAPK/ERK signaling pathway by preventing RAF-dependent MEK phosphorylation and suppressing ERK activation to inhibit tumor cell proliferation, migration, and induce apoptosis.

Primary Applications and Mechanism of Action