Niraparib is a potent PARP1/2 inhibitor. It affects DDR signaling by trapping PARP at DNA breaks to inhibit tumor cell growth.
Comprehensive IC50 Values for Niraparib (MK-4827) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Niraparib is a potent PARP1/2 inhibitor. It affects DDR signaling by trapping PARP at DNA breaks to inhibit tumor cell growth.