Darovasertib (LXS196) is a potent, selective PKC inhibitor. It affects PKC signaling, by blocking kinase activity, inhibiting uveal melanoma (UM) progression, and is safely evaluated in combination with crizotinib.
Comprehensive IC50 Values for Darovasertib (LXS196) Across Cell-free Enzyme Inhibitory Profiles and Cell-based Functional Assays.
Darovasertib (LXS196) is a potent, selective PKC inhibitor. It affects PKC signaling, by blocking kinase activity, inhibiting uveal melanoma (UM) progression, and is safely evaluated in combination with crizotinib.