3-Deazaneplanocin A (DZNep) Hydrochloride Mechanism of Action: EZH2 Inhibition in Cancer Cell Research

3-Deazaneplanocin A (DZNep) Hydrochloride MOA:Targeting EZH2/PRC2 Pathway for Oncology and Cancer Epigenetics

🎯 check 3-Deazaneplanocin A (DZNep) Hydrochloride product page

3-Deazaneplanocin A (DZNep) Hydrochloride is a potent, dose-dependent EZH2 and histone methyltransferase inhibitor. It affects Wnt/β-catenin, PTEN/Akt, and NF-κB signaling pathways by reducing H3K27 trimethylation (H3K27me3) and modulating gene transcription, effectively inhibiting cancer cell proliferation and fibrosis while promoting apoptosis and differentiation.

Primary Applications and Mechanism of Action