Tianeptine sodium

Catalog No.S1436

Tianeptine sodium is a selective serotonin reuptake enhancer (SSRE) compound used for treating major depressive episodes.

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In DMSO USD 130 In stock
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Tianeptine sodium Chemical Structure

Tianeptine sodium Chemical Structure
Molecular Weight: 458.93

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Related Compound Libraries

Tianeptine sodium is available in the following compound libraries:

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Product Description

Biological Activity

Tianeptine (INN) (Stablon, Coaxil, Tatinol) is a selective serotonin reuptake enhancer (SSRE) drug used for treating major depressive episodes (mild, moderate, or severe). Unlike conventional tricyclic antidepressants, tianeptine enhances the reuptake of serotonin instead of inhibiting it, opposite to the action of SSRIs. Moreover, it enhances the extracellular concentration of dopamine in the nucleus accumbens and modulates the D2 and D3 dopamine receptors. There is also action on the NMDA and AMPA receptors. [1]

Chemical Information

Download Tianeptine sodium SDF
Molecular Weight (MW) 458.93
Formula

C21H24ClN2NaO4S

CAS No. 30123-17-2
Storage 3 years -20℃Powder
6 months-80℃in DMSO
Synonyms
Solubility (25°C) * In vitro DMSO 92 mg/mL (200 mM)
Water 92 mg/mL (200 mM)
Ethanol 92 mg/mL (200 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Selleck tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Chemical Name Heptanoic acid, 7-[(3-chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino]-, sodium salt (1:1)

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