E
E
E
E
L
L
C
C
C
C
C
C
C
C
C
C
C
F
F
F
F
F
F
F
F
F
F
F
F
F
F
F
F
F
A
A
F
Kinase
Fibronetin
Cysteine Rich
Leucine Rich
EGF-Like
Acid Box
Cadherin
IG-Like
Glycine Rich
EGFR
HER2/ErbB2
ErbB3
ErbB4
INSR
IGF-1R
IRR
FGFR
PDGFR
CSF-1R
Kit
FLT3
VEGFR
Met
Ron
Sea
TrkA
TrkB
TrkC
Tie
Tie-2
Eph
Eck
Eek
Erk
Elk
Ros
Ret
Ltk
ALK
PLC
PDK-1
Akt
PKC
IKK
Syk
Bcr-Abl
Ras
Raf
c-Src
GSK-3
c-Jun
c-Fos
JA
K
R
O
C
K
R
ho
P
A
K
JA
K
S
T
A
T
PI3K/Akt
Pathway
NF-κB
Pathway
MAPK
Pathway
Cell Cycle
JAK/STAT
Pathway
Ⅰ
Ⅱ
Ⅲ
Ⅳ
Ⅴ
Ⅵ
Ⅶ
HER2/ErbB2 Inhibitors
CP-724714
Afatinib
Dacomitinib
Pan-EGFR Inhibitors
Afatinib
Lapatinib
Sapitinib
Selective EGFR Inhibitors
Erlotinib (EGFR/ErbB1)
CP-724714 (HER2/ErbB2)
Mutant EGFR Inhibitors
Osimertinib
Gefitinib
Pan-FGFR Inhibitors
BGJ398
AZD4547
Erdafitinib
Selective FGFR Inhibitors
PD173074
(
FGFR1
)
H3B-6527
(
FGFR4
)
Pan-PDGFR Inhibitors
Imatinib
Crenolanib
CP-673451
Selective PDGFR Inhibitors
Sunitinib (PDGFRβ)
Avapritinib (PDGFRα)
c-Kit Inhibitors
Sitravatinib
Masitinib
Amuvatinib
Dovitinib
Pan-VEGFR Inhibitors
Axitinib
Regorafenib
Nintedanib
Lenvatinib
Selective VEGFR Inhibitors
Cabozantinib (VEGFR2)
Anlotinib (VEGFR2)
SAR131675 (VEGFR3)
Tie-2 Inhibitors
Tie2 kinase Inhibitor
Cabozantinib
c-RET Inhibitors
AD80
GSK3179106
ALK Inhibitors
Brigatinib
Ceritinib
Lorlatinib
Alectinib
Repotrectinib
IGF-1R Inhibitors
Linsitinib
GSK1904529A
BMS-754807
Picropodophyllin
c-Met Inhibitors
Crizotinib (PF-02341066)
Capmatinib
Foretinib
BMS-777607
PHA-665752
Savolitinib
Pan-Trk Inhibitors
Larotrectinib
Entrectinib
Selitrectinib
Selective Trk Antagonist
ANA-12 (TrkB)
Selective Trk Agonist
7,8-Dihydroxyflavone (TrkB)
P
Cell Cycle
MAPK
Pathway
PI3K/Akt
Pathway
NF-κB
Pathway
JAK/STAT
Pathway
Kinase
Fibronetin
Cysteine Rich
Leucine Rich
EGF-Like
Acid Box
Cadherin
IG-Like
Glycine Rich
Tie
Eph
Eck
Eek
Erk
Elk
Ros
Ltk
Sea
IRR
I
II
III
IV
V
VI
VII
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Notes:
1:Clickable
2:Unclickable