• PAK1
  • PAK3
  • PAK2
  • PAK4
  • PAK5
  • PAK6

PAK6 Inhibitors

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S7094 PF-3758309 PF-03758309 (PF-03758309) is a potent, ATP-competitive, pyrrolopyrazole inhibitor of PAK4 with Kd of 2.7 nM. PF-3758309 is antiproliferative and induces apoptosis in a HCT116 tumor model. Pan PAK6, Ki: 17.1 nM