P2Y receptor Selective Inhibitors | Antagonists
| Catalog No. | Product Name | Information | Selective / Pan | IC50 / Ki |
|---|---|---|---|---|
| S4079 | Ticagrelor | Ticagrelor is the first reversibly binding oral P2Y12 receptor antagonist with Ki of 2 nM. |
Selective | P2Y12, Ki: 2 nM |
| S2855 | MRS 2578 | MRS2578 is a potent P2Y6 receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors. |
Selective | P2Y6, IC50: 37 nM |
| S1415 | Clopidogrel | Clopidogrel is an oral, thienopyridine class antiplatelet agent. |
Selective | |
| S1258 | Prasugrel | Prasugrel is a thienopyridine ADP receptor (P2Y12) antagonist, used for the reduction of thrombotic cardiovascular events. |
Selective |
