D4 receptor Agonists | Antagonists
| Catalog No. | Product Name | Information | Selective / Pan | IC50 / Ki |
|---|---|---|---|---|
| S2011 | Pramipexole 2HCl Monohydrate | Pramipexole 2HCl Monohydrate is a partial/full D2S, D2L, D3, D4, receptor agonist with a Ki of 3.9, 2.2, 0.5, 5.1 nM. |
Pan | D4 receptor, Ki: 5.1 nM |
| S2460 | Pramipexole | Pramipexole is a partial/full D2S, D2L, D3, D4 receptor agonist with a Ki of 3.9, 2.2, 0.5 and 5.1 nM for D2S, D2L, D3, D4 receptor, respectively. |
Pan | D4 receptor, Ki: 5.1 nM |
| S4086 | Loxapine Succinate | Loxapine Succinate is a D2DR and D4DR inhibitor, serotonergic receptor antagonist and also a dibenzoxazepine anti-psychotic agent. |
Pan | D4 receptor (human), Ki: 7.5 nM |
