CXCR4 Selective Antagonists

Catalog No. Product Name Information Selective / Pan IC50 / Ki
S2912 WZ811

WZ811 is a highly potent competitive CXCR4 antagonist with EC50 of 0.3 nM.

Selective CXCR4, EC50: 0.3 nM
S8030 Plerixafor (AMD3100)

Plerixafor is a chemokine receptor antagonist for CXCR4 and CXCL12-mediated chemotaxis with IC50 of 44 nM and 5.7 nM, respectively.

Selective CXCR4, IC50: 44 nM
S3013 Plerixafor 8HCl (AMD3100 8HCl)

Plerixafor 8HCl (AMD3100 8HCl) is the hydrochloride of Plerixafor, a chemokine receptor antagonist for CXCR4 and CXCL12-mediated chemotaxis with IC50 of 44 nM and 5.7 nM, respectively.

Selective CXCR4, IC50: 44 nM