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Inflammation

Cat.No.	Product Name	Added

S1634	Acetaminophen	Oct 2010
Acetaminophen is a highly selective inhibitor of COX-2 and 6-keto-PGF1 alpha with IC50 of 302.3 mg/kg and 10 µM, respectively.

S1368	Acitretin	Jul 2010
Acitretin is a second generation retinoid used for psoriasis.

S1647	Adenosine(Adenocard)	Oct 2010
Adenosine is a nucleoside composed of a molecule of adenine attached to a ribose sugar molecule (ribofuranose) moiety via a β-N9-glycosidic bond.

S1139	ADL5859	Jan 2010
ADL-5859 is an δ-opioid receptor agonist (Ki=0.84 nM, EC50=20 nM).

S2258	Aesculin(Esculin)	Dec 2010
Aesculin(Esculin) is a glucoside found in horse chestnuts.

S2552	Azelastine	May 2011
Azelastine is a potent, second-generation, selective, histamine antagonist.

S1500	Betamethasone (Celestone)	Sep 2010
Betamethasone is a glucocorticoid steroid with anti-inflammatory and immunosuppressive properties.

S1688	Betamethasone Dipropionate(Diprolene)	Dec 2010
Betamethasone Dipropionate(Diprolene) is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities.

S1690	Betamethasone valerate (Betnovate, Celestone)	Dec 2010
Betamethasone valerate(Betnovate, Celestone) is a moderately potent glucocorticoid steroid with anti-inflammatory and immunosuppressive properties.

S1689	Betapar(Meprednisone)	Dec 2010
Betapar(Meprednisone) is a glucocorticoid and a methylated derivative of prednisone.

S1574	BIRB 796 (Doramapimod)	Nov 2010
BIRB 796 (Doramapimod) a small molecule of p38 MAPK inhibitor with Kd of 0.1 nM is available at Selleck.

S1286	Budesonide	Jun 2010
Budesonide is a glucocorticoid steroid for the treatment of asthma, non-infectious rhinitis.

S1290	Celastrol	Jun 2010
Celastrol, a plant-derived triterpene, has anti-inflammatory and immunosuppressive activity.

S1261	Celecoxib	May 2010
COX-2 inhibitor,IC50=0.04uM

S1291	Cetirizine di hcl	Jun 2010
Cetirizine is an antihistamine.

S1292	Chelerythrine Chloride	Jun 2010
Chelerythrine is a potent, selective, and cell-permeable PKC inhibitor (IC50 = 660 nM).

S1677	Chloramphenicol(Chloromycetin)	Dec 2010
Chloramphenicol(Chloromycetin) is a bacteriostatic antimicrobial.

S1839	Chloroxine	Nov 2010
Chloroxine is a synthetic antibacterial compound that is effective in the treatment of dandruff and seborrheic dermatitis when incorporated in a shampoo.

S1816	Chlorpheniramine	Jan 2011
Chlorpheniramine, a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.

S2281	Chrysin	Jan 2011
Chrysin is a naturally occurring flavone chemically extracted from the blue passion flower (Passiflora caerulea).

S1845	Cimetidine (Tagamet)	Dec 2010
Cimetidine (Tagamet), a histamine congener, competitively inhibits histamine binding to histamine H2 receptors.

S2559	Cortisone acetate (Cortone)	May 2011
Cortisone acetate (Cortone) is an acetate salt form of cortisone that is a steroid hormone and a glucocorticoid.

S1888	Deflazacort(Calcort)	Oct 2010
Deflazacort(Calcort) is a glucocorticoid used as an anti-inflammatory and immunosuppressant.

S1701	Desonide	Dec 2010
Desonide is a low potency topical corticosteroid.

S1322	Dexamethasone	Jun 2010
Dexamethasone is an anti-inflammatory and immunosuppressant.

S1903	Diclofenac	Jan 2011
Diclofenac is a non-selective COX inhibitor with IC50 of 60 and 220 nM for ovine COX-1 and -2, respectively.

S1858	Dienestrol(Restrol)	Jan 2011
Dienestrol(Restrol) is a synthetic, non-steroidal estrogen. It is an estrogen receptor agonist.

S1866	Diphenhydramine (Benadryl)	Dec 2010
Diphenhydramine (Benadryl), a histamine H1 antagonist used as an antiemetic, antitussive, for dermatoses and pruritus, for hypersensitivity reactions, as a hypnotic, an antiparkinson, and as an ingredient in common cold preparations.

S2295	Emodin	Jan 2011
Emodin is a purgative resin, 6-methyl-1,3,8-trihydroxyanthraquinone, from rhubarb, the buckthorn and Japanese Knotweed (Fallopia japonica).

S1743	Esomeprazole magnesium(Nexium)	Jan 2011
Esomeprazole magnesium(Nexium) is a proton pump inhibitor to reduce gastric acid secretion.

S1328	Etodolac(Lodine)	Jun 2010
Etodolac (Lodine SR, Eccoxolac) is a COX inhibitor with an IC50 of 53.5 nM.

S2298	Fisetin (Fustel)	Jan 2011
Fisetin (Fustel) is a potent sirtuin activating compound (STAC) and an agent that modulates sirtuins.

S1513	Flunisolide (Nasalide)	Sep 2010
Flunisolide (AeroBid, Nasalide, Nasarel) is a corticosteroid often prescribed as treatment for allergic rhinitis.

S2608	Fluocinonide(Vanos)	Sep 2010
Fluocinonide(Vanos) is a potent glucocorticoid steroid used topically as anti-inflammatory agent for the treatment of skin disorders such as eczema.

S1679	Flurbiprofen(Ansaid)	Jan 2011
Flurbiprofen is a member of the phenylalkanoic acid derivative family of non-steroidal anti-inflammatory drugs (NSAIDs).

S2129	Fudosteine	Jan 2011
Fudosteine is a novel mucoactive agent and a MUC5AC mucin hypersecretion inhibitor.

S2302	Glycyrrhizic acid	Jan 2011
Glycyrrhizic acid is a widely used anti-inflammatory agent isolated from the licorice root.

S2309	Hesperidin	Jan 2011
Hesperidin is a flavanone glycoside found abundantly in citrus fruits.

S1638	Ibuprofen (Advil)	Oct 2010
Ibuprofen (Advil) is a non-selective COX inhibitor with an IC50 of 0.33 mM.

S1518	Ibuprofen Lysine (NeoProfen)	Sep 2010
Ibuprofen Lysine (NeoProfen) is a non-steroidal anti-inflammatory agent.

S2534	Isoconazole nitrate (Travogen)	Apr 2011
Isoconazole nitrate (Travogen) is an azole antifungal reagent.

S2170	ITF2357 (Givinostat)	Jan 2011
ITF2357 (Givinostat) is a noverl HDAC inhibitor with IC50 of 10, 7.5 and 16 nM for maize HDAC preparations HD2, HD-1B and HD-1A, respectively.

S1645	Ketoprofen (Actron)	Oct 2010
Ketoprofen (Actron) is a non-selective NSAID with IC50 of 0.5 μM and 2.33 μM for human recombinant COX-1 and COX-2, respectively.

S1646	Ketorolac (Toradol)	Oct 2010
Ketorolac (Toradol) is a non-selective COX inhibitor with IC50 of 31.5 µM and 60.5 µM for human recombinant COX-1 and COX-2, respectively.

S1706	Lamivudine(Epivir)	Dec 2010
Lamivudine(Epivir) is a potent nucleoside analog reverse transcriptase inhibitor with an IC50 of 2.7 mM.

S1354	Lansoprazole	Jun 2010
Lansoprazole is a proton-pump inhibitor (PPI) which prevents the stomach from producing gastric acid.

S2387	Lappaconite Hydrobromide	Feb 2011
Lappaconite Hydrobromide is a kind of alkaloid extracted from Aconitum sinomontanum Nakai and has anti-inflammatory effects.

S1247	Leflunomide	May 2010
Immunosuppressant agent. Its active metabolite is A77 1726 (RS-61980).

S1939	Levamisole Hydrochloride(Ergamisol)	Dec 2010
Levamisole Hydrochloride(Ergamisol)is an antihelminthic drug that has been tried experimentally in rheumatic disorders where it apparently restores the immune response by increasing macrophage chemotaxis and T-lymphocyte function.

S2319	Limonin	Jan 2011
Limonin is also known as limonoate D-ring-lactone and limonoic acid di-delta-lactone. Chemically, it is a member of the class of compounds known as furanolactones.

S1358	Loratadine	Jun 2010
Loratadine is a selective inverse peripheral histamine H1-receptor agonist with an IC50 of >32 μM.

S1669	Loteprednol etabonate	Dec 2010
Loteprednol etabonate is an anti-inflammatory corticosteroid used in ophthalmology

S2320	Luteolin	Jan 2011
Luteolin is a PDE4 inhibitor and a general phosphodiesterase inhibitor, and an Interleukin 6 inhibitor.

S1110	LY315920(Varespladib)	Sep 2009
LY315920 (Varespladib) is a sPLA2 inhibitor (IC50 of 9.6 ±1 nM).

S1137	Malotilate	Dec 2009
Malotilate is a liver protein metabolism improved compound.

S1734	Meloxicam (Mobic)	Jan 2011
Meloxicam (Mobic) is a nonsteroidal anti-inflammatory agent with analgesic and fever reducer effects.

S1681	Mesalamine (Lialda, Apriso)	Nov 2010
Mesalamine (Lialda, Apriso) is an anti-inflammatory compound.

S2323	Methyl-Hesperidin	Jan 2011
Methyl-Hesperidin is a flavanone glycoside (flavonoid) (C28H34O15) found abundantly in citrus fruits. Its aglycone form is called hesperetin.

S1733	Methylprednisolone	Dec 2010
Methylprednisolone is a synthetic corticosteroid with anti-inflammatory and immunomodulating properties.

S1987	Mometasone furoate	Jan 2012
Mometasone furoate is a glucocorticosteroid used topically to reduce inflammation of the skin or in the airways.

S2327	Myricitrin(Myricitrine)	Jan 2011
Myricitrin(Myricitrine) is a chemical compound. It can be isolated from the root bark of Myrica cerifera (Bayberry, a small tree native to North America) and in Chrysobalanus icaco.

S1626	Naproxen (Aleve)	Oct 2010
Naproxen (Aleve) is a non-selective cyclooxygenase (COX) inhibitor with IC50 of 8.7 Â± 0.23 mg/kg.

S1255	Nepafenac	May 2010
Nepafenac is a non-steroidal anti-inflammatory agent.

S1971	Nicorandil(Ikorel)	Dec 2010
Nicorandil(Ikorel) is potassium channel activator.

S1899	Nicotinamide (Niacinamide)	Dec 2010
Nicotinamide(Niacinamide) is a water-soluble vitamin and is part of the vitamin B group.

S2334	Oleanolic Acid(Caryophyllin)	Jan 2011
Oleanolic acid(Caryophyllin) is a naturally occurring triterpenoid, widely distributed in food and medicinal plants, related to betulinic acid. It is relatively non-toxic, antitumor, and hepatoprotective, as well as exhibiting antiviral. properties.

S2339	Paeonol (Peonol)	Jan 2011
Paeonol(Peonol) is a major component extracted from Chinese herbs moutan cortex and Cynanchum paniculatum .

S2397	Palmatine chloride	Mar 2011
Palmatine hydrochloride (Palmatine chloride (6CI,7CI); Fibrauretin) is a hydrochloride salt of palmatine which is a protoberberine alkaloid.

S2341	Parthenolide ((-)-Parthenolide)	Jan 2011
Parthenolide ((-)-Parthenolide) is a sesquiterpene lactone which occurs naturally in the plant feverfew (Tanacetum parthenium).

S2666	PF-3845	Sep 2011
PF-3845 is a potent, selective and irreversible fatty acid amide hydrolase (FAAH) inhibitor with a Ki of 0.23 μM.

S1654	Phenylbutazone(Butazolidin, Butatron)	Dec 2010
Phenylbutazone(Butazolidin, Butatron) is used as a non-steroidal anti-inflammatory agent for the treatment of chronic pain, including the symptoms of arthritis.

S2342	Phloretin(Dihydronaringenin)	Jan 2011
Phloretin(Dihydronaringenin) is a dihydrochalcone, a type of polyphenol.

S5004	Pimecrolimus	Apr 2009
Pimecrolimus is an inhibitor of inflammatory cytokine secretion

S1713	Piroxicam (Feldene)	Dec 2010
Piroxicam (Feldene) is a non-selective COX inhibitor with an IC50 of 6 mM.

S1588	Pravadoline(WIN 48098)	Nov 2010
Pravadoline (WIN 48098) is an antiinflammatory and analgesic compound with an IC50 of 4.9 µM for inhibition of the synthesis of prostaglandins (PGs) in mouse brain.

S2570	Prednisolone acetate (Omnipred)	May 2011
Prednisolone acetate is a synthetic corticosteroid drug that is particularly effective as an immunosuppressant agent.

S1737	Prednisolone(Hydroretrocortine)	Dec 2010
Prednisolone(Hydroretrocortine) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.

S1622	Prednisone(Adasone)	Dec 2010
Prednisone (Deltasone, Liquid Pred, Orasone, Adasone) is a synthetic corticosteroid agent that is particularly effective as an immunosuppressant compound.

S6003	PTC124 (Ataluren)	Apr 2009
PTC124 also known as Ataluren is CFTR-G542X nonsense allele inhibitor.

S2347	Quercetin dihydrate(Sophoretin)	Jan 2011
Quercetin, a flavonol widely distributed in plants. It is an antioxidant, like many other phenolic heterocyclic compounds.

S2391	Quercetin(Sophoretin)	Feb 2011
Quercetin is a PI3K and PKC inhibitor with IC50 of 3.8 μM and 15µg/ml.

S2032	Rebamipide	Jan 2012


S1396	Resveratrol	Jul 2010
Resveratrol is a phytoalexin produced naturally by several plants with anti-cancer, anti-inflammatory, blood-sugar-lowering and other beneficial cardiovascular effects .

S2395	Rheochrysidin(Physcione)	Mar 2011
Rheochrysidin (Physcion; physcione; parietin) is one of the major components of Da-Cheng-Qi decoction used in the treatment of inflammation.

S2131	Roflumilast(Daxas)	Jan 2011
Roflumilast(Daxas) is a selective, long-acting the enzyme PDE-4 inhibitor with an IC50 of 0.8 nM.

S1430	Rolipram	Jul 2010
Rolipram is a PDE4-inhibitor and an anti-inflammatory agent.

S2556	Rosiglitazone (Avandia)	May 2011
Rosiglitazone (Avandia) is a potent antihyperglycemic agent and a potent thiazolidinedione insulin sensitizer with IC50 of 12, 4 and 9 nM for rat, 3T3-L1 and human adipocytes, respectively.

S2349	Rutaecarpine(Rutecarpine)	Jan 2011
Rutaecarpine is an indolopyridoquinazolinone alkaloid isolated from Evodia rutaecarpa and related herbs.

S2127	S-(+)-Rolipram	Jan 2011
S-(+)-Rolipram is a less active enantiomer of the PDE4 inhibitor with an EC50 of 1.0 µM.

S2351	Salicin(Salicoside, Salicine)	Jan 2011
Salicin(Salicoside, Salicine) is an alcoholic β-glycoside that contains D-glucose. Salicin is an anti-inflammatory agent that is produced from willow bark.

S1077	SB 202190	Jun 2009
P38 MAP(mitogen activated protein) Kinase inhibitor.

S1076	SB 203580	Jun 2009
SB 203580 is a potent inhibitor of LPS-induced cytokine synthesis in the human monocyte cell line THP-1 (IC50 = 50-100 nM).

S2359	Sinomenine(Cucoline)	Jan 2011
Sinomenine(Cucoline) is traditionally used in herbal medicine in these countries, as a treatment for rheumatism and arthritis.

S2007	Sulindac(Clinoril)	Dec 2010
Sulindac(Clinoril) is a non-steroidal anti-inflammatory agent of the arylalkanoic acid class.

S1569	Tazarotene(Avage)	Nov 2010
Tazarotene is a prescription topical retinoid sold as a cream or gel.

S1984	Ticlopidine hydrochloride	Jan 2012
Ticlopidine hydrochloride is a hydrochloride salt form of ticlopidine which is selective P2Y12 receptor antagonist. Inhibits ADP-induced platelet aggregation and displays antithrombotic activity following oral administration in vivo.

S1628	Triamcinolone Acetonide	Oct 2010
Triamcinolone Acetonide is a more potent type of triamcinolone, being about 8 times as effective as prednisone.

S1933	Triamcinolone(Aristocort)	Dec 2010
Triamcinolone(Aristocort) is a glucocorticoid given, as the free alcohol or in esterified form, orally, intramuscularly, by local injection, by inhalation, or applied topically in the management of various disorders in which corticosteroids are indicated.

S1168	Valproate	Mar 2010
Valproate is a histone deacetylase inhibitor with an IC50 of 0.4 mM and exhibits anticancer, anti-inflammatory and neuroprotective effects.

S1458	VX-745	Aug 2010
VX-745 is a lead anti-inflammatory candidate, p38 MAPK inhibitor (IC50=10 nM) for the treatment of Rheumatoid arthritis (RA).