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Immunology

Cat.No.	Product Name	Added

S1210	Abitrexate(Methotrexate)	May 2010
Abitrexate(Methotrexate) is an antimetabolite and antifolate agent with antineoplastic and immunosuppressant activities.

S2189	Acitazanolast	Jan 2011
Acitazanolast is an active metabolite of tazanolast and anti-allergic drug.

S2204	Atazanavir sulfate	Mar 2011
Atazanavir sulfate(BMS-232632-05) is a sulfate salt form of atazanavir (BMS-232632) that is an highly potent HIV protease inhibitor with EC50 and EC90 of 2.6~5.3 nM and 9~15 nM in cell culture.

S1721	Azathioprine(Azasan, Imuran)	Jan 2011
Azathioprine(Azasan, Imuran) is a drug that suppresses the immune system and is used in organ transplantation and autoimmune disease.

S2270	Bergenin (Cuscutin)	Dec 2010
Bergenin (Cuscutin) is trihydroxybenzoic acid glycoside and the C-glycoside of 4-O-methyl gallic acid.

S1500	Betamethasone (Celestone)	Sep 2010
Betamethasone is a glucocorticoid steroid with anti-inflammatory and immunosuppressive properties.

S1688	Betamethasone Dipropionate(Diprolene)	Dec 2010
Betamethasone Dipropionate(Diprolene) is a glucocorticoid steroid with anti-inflammatory and immunosuppressive abilities.

S1290	Celastrol	Jun 2010
Celastrol, a plant-derived triterpene, has anti-inflammatory and immunosuppressive activity.

S2280	Chlorogenic acid	Jan 2011
Chlorogenic acid is a hydroxycinnamic acid and a member of a family of naturally occurring organic compounds.

S1816	Chlorpheniramine	Jan 2011
Chlorpheniramine, a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.

S2416	Chondroitin sulfate	Sep 2011
Chondroitin sulfate is a kind of sulfated glycosaminoglycan (GAG) which is composed of a chain of alternating sugars including N-acetylgalactosamine and glucuronic acid.

S1847	Clemastine Fumarate	Dec 2010
Clemastine fumarate, a histamine H1 antagonist used as the hydrogen fumarate in hay fever, rhinitis, allergic skin conditions, and pruritus.

S2559	Cortisone acetate (Cortone)	May 2011
Cortisone acetate (Cortone) is an acetate salt form of cortisone that is a steroid hormone and a glucocorticoid.

S2286	Cyclosporin A(Cyclosporine A)	Jan 2011
Cyclosporin A (cyclosporine, cyclosporin ) is an immunosuppressant agent widely used in post-allogeneic organ transplant to reduce the activity of the immune system.

S1514	Cyclosporine (Neoral)	Dec 2010
Cyclosporine (Neoral) is an immunosuppressant drug.

S1888	Deflazacort(Calcort)	Oct 2010
Deflazacort(Calcort) is a glucocorticoid used as an anti-inflammatory and immunosuppressant.

S1866	Diphenhydramine (Benadryl)	Dec 2010
Diphenhydramine (Benadryl), a histamine H1 antagonist used as an antiemetic, antitussive, for dermatoses and pruritus, for hypersensitivity reactions, as a hypnotic, an antiparkinson, and as an ingredient in common cold preparations.

S2293	DL-Carnitine hydrochloride	Jan 2011
DL-Carnitine hydrochloride is a quaternary ammonium compound biosynthesized from the amino acids lysine and methionine.

S1504	Dyphylline(Dilor)	Sep 2010
Dyphylline(Dilor, Lufyllin, diprophylline) is a xanthine derivative with bronchodilator and vasodilator effects.

S2229	Eltrombopag (SB-497115-GR)	Apr 2011
Eltrombopag (SB-497115-GR, Promacta, Revolade) is a small molecule agonist of the c-mpl (TpoR) receptor with an IC50 of 0.69 μM for the inhibition of hERG K+ channel tail current.

S1704	Emtricitabine (Emtriva)	Jan 2011
Emtricitabine (Emtriva) is a nucleoside reverse transcriptase inhibitor with an IC50 of 27.7 μM.

S1743	Esomeprazole magnesium(Nexium)	Jan 2011
Esomeprazole magnesium(Nexium) is a proton pump inhibitor to reduce gastric acid secretion.

S5003	FK-506 (Tacrolimus)	Apr 2009
A immunosuppressive agent and macrolide antibiotic.

S1331	Fluconazole	Jun 2010
Fluconazole is a triazole antifungal drug used in the treatment and prevention of superficial and systemic fungal infections.

S1992	Fluticasone propionate (Flonase, Veramyst)	Jan 2012
Fluticasone propionate (Flonase, Veramyst) is a synthetic corticosteroid which is derived from fluticasone used to treat asthma and allergic rhinitis (hay fever).

S2625	Fostamatinib disodium (R788)	May 2011
Fostamatinib disodium (R788) is an important spleen tyrosine kinase (Syk) inhibitor and a free base of R788 (FosD, fostamatinib disodium, tamatinib fosdium) which is also a selective Syk inhibitor with an IC50 of 41 nM.

S5002	FTY720(Fingolimod)	Apr 2009
FTY720 Fingolimod Gilenia is Src-bcr-Abl Inhibitor & S1P receptor agonist with IC50 of 0.137, 10.98 nM for (S)- and (R)- FTY720-phosphate.

S1343	Ginkgolide B	Jun 2010
The ginkgolide B is a platelet-activating factor (PAF) receptor antagonist (Ki = 1.3 μM)

S2149	GSK1292263	Dec 2010
GSK1292263 is a novel GPR119 receptor agonist used for the treatment of type 2 diabetes.

S1211	Imiquimod	May 2010
Imiquimod(Aldara) is a novel synthetic agent with immune response modifying activity.

S2483	Metformin(Glucophage)	Jan 2011
Metformin(Glucophage) is an AMP-activated protein kinase agonist.

S1733	Methylprednisolone	Dec 2010
Methylprednisolone is a synthetic corticosteroid with anti-inflammatory and immunomodulating properties.

S1501	Mycophenolate mofetil (CellCept)	Sep 2010
Mycophenolate mofetil is a inhibitor of inosine monophosphate dehydrogenase and a immunosuppressant.

S2487	Mycophenolic acid(Mycophenolate)	Jan 2011
Mycophenolic acid (mycophenolate) is an immunosuppressant agent used to prevent rejection in organ transplantation.

S2489	Nateglinide(Starlix)	Jan 2011
Nateglinide(Starlix) is an insulin secretagog agent that lowers blood glucose levels by stimulating insulin secretion from the pancreas.

S2494	Olopatadine hydrochloride(Opatanol)	Jan 2011
Olopatadine hydrochloride(Opatanol) is a histamine blocker and mast cell stabilizer with an IC50 of 559 µM for the release of histamine.

S2338	Oxymatrine(Matrine N-oxide)	Jan 2011
Oxymatrine(Matrine N-oxide) is one of components of the root of Sophora flavescens.

S2339	Paeonol (Peonol)	Jan 2011
Paeonol(Peonol) is a major component extracted from Chinese herbs moutan cortex and Cynanchum paniculatum .

S2542	Phenformin hydrochloride	Apr 2011
Phenformin hydrochloride is a hydrochloride salt of phenformin that is an anti-diabetic drug from the biguanide class.

S1921	Phenindione(Rectadione)	Dec 2010
Phenindione is an anticoagulant which functions as a Vitamin K antagonist.

S1567	Pomalidomide	Nov 2010
Pomalidomide is tumor necrosis factor-α inhibitor and a new immunomodulator with an IC50 of 1 μM.

S1622	Prednisone(Adasone)	Dec 2010
Prednisone (Deltasone, Liquid Pred, Orasone, Adasone) is a synthetic corticosteroid agent that is particularly effective as an immunosuppressant compound.

S1988	Propylthiouracil	Dec 2010
Propylthiouracil is a thyroperoxidase and 5'-deiodinase inhibitor.

S2194	R406	Jan 2011
R406 is an orally available spleen tyrosine kinase inhibitor with an IC50 of 41 nM.

S2206	R935788 (Fostamatinib)	Mar 2011
R935788 (Fostamatinib) is a selective Syk inhibitor with an IC50 of 41 nM.

S2400	Rhein(Monorhein)	Mar 2011
Rhein(Monorhein; NSC 38629; Rheic acid; Rheinic acid) is a constituent of rhubarb which was isolated from the fresh rhizome of Rheum coreanum Nakai.

S2556	Rosiglitazone (Avandia)	May 2011
Rosiglitazone (Avandia) is a potent antihyperglycemic agent and a potent thiazolidinedione insulin sensitizer with IC50 of 12, 4 and 9 nM for rat, 3T3-L1 and human adipocytes, respectively.

S2505	Rosiglitazone maleate	Jan 2011
Rosiglitazone maleate (Avandia) is an anti-diabetic agent in the thiazolidinedione class of agents.

S2359	Sinomenine(Cucoline)	Jan 2011
Sinomenine(Cucoline) is traditionally used in herbal medicine in these countries, as a treatment for rheumatism and arthritis.

S1433	Suplatast tosylate	Jul 2010
Suplatast tosilate is a Th2 cytokine inhibitor which is used as an antiallergic drug.

S2403	Tetrandrine(Fanchinine)	Mar 2011
Tetrandrine (Fanchinine; Hanfangchin A) is a calcium channel blocker with an IC50 of 38.23± 25.77 μM.

S1193	Thalidomide	Apr 2010
Thalidomide was introduced as a sedative agent, immunomodulatory agent and also is investigated for treating symptoms of many cancers.

S1621	Theophylline(Theo-Dur)	Oct 2010
Theophylline (Theo-Dur) is a methylxanthine agent and has bronchodilator properties and is used in the treatment of asthma and COAD.

S1774	Thioguanine	Dec 2010
Thioguanine (6-Thioguanine) is a purine antimetabolite widely used in the treatment of acute lymphoblastic leukemia, autoimmune disorders (e.g., Crohn's disease, rheumatoid arthritis) and organ transplant recipients.

S5001	Tofacitinib (CP-690550)	Apr 2009
Tofacitinib (CP-690550) is a novel, small molecule potent and selective JAK-3 kinase inhibitor with an IC50 of 1 nM for inhibition of the JAK-3 activities.

S1439	Tranilast(SB 252218)	Jul 2010
Tranilast (Rizaben) is an antiallergic compound.

S2022	Trioxsalen(Trisoralen)	Jan 2011
Trioxsalen(Trisoralen) is a furanocoumarin and a psoralen derivative.

S6005	VX-702	Apr 2009
VX-702 is a P38 MAPK inhibitor , IL-6, IL-1β and TNFα (IC50 = 59, 122 and 99 ng/ml, respectively)

S2228	VX-765	Apr 2011
VX-765 is a novel and irreversible IL-converting enzyme/caspase-1 inhibitor with an IC50 of 0.8 nM.

S1565	VX-809	Nov 2010
VX-809 is the second investigational oral candidate compound for the treatment of cystic fibrosis (CF).

S1633	Zafirlukast(Accolate)	Oct 2010
Zafirlukast is a leukotriene receptor antagonist (LTRA). (IC50=0.6μM, IC50=7.0 µM for CYP2C9)

S1443	Zileuton	Jul 2010
Zileuton (ZYFLO) is an orally active inhibitor of 5-lipoxygenase, and thus inhibits leukotrienes (LTB4, LTC4, LTD4, and LTE4) formation.