Home GPCR & G Protein CCK receptor inhibitor Rebamipide For research use only.

Rebamipide

Synonyms: OPC-12759,Proamipide

Rebamipide (OPC-12759,Proamipide) is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [125I]BH-CCK-8S with IC50 of 37.7 μM.

Rebamipide Chemical Structure

Rebamipide Chemical Structure

CAS: 90098-04-7

Selleck's Rebamipide has been cited by 2 publications

Purity & Quality Control

Batch: S203201 DMSO] 74 mg/mL] false] Water] Insoluble] false] Ethanol] Insoluble] false Purity: 99.97%
99.97

Rebamipide Related Products

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Biological Activity

Description Rebamipide (OPC-12759,Proamipide) is a cholecystokinin type 1 (CCK1) receptor inhibitor for inhibiting [125I]BH-CCK-8S with IC50 of 37.7 μM.
NCT Number Recruitment Conditions Sponsor/Collaborators Start Date Phases
NCT04150172 Completed
Healthy Volunteers
Korea Otsuka Pharmaceutical Co. Ltd.
 April 22 2019 Phase 1
NCT02106130 Completed
Healthy
IlDong Pharmaceutical Co Ltd
 May 2013 Phase 1
NCT01167101 Completed
Stomach Ulcer
Kangdong Sacred Heart Hospital
 May 2009 Not Applicable
NCT00997789 Completed
Therapeutic Equivalency|Pharmacogenetics
Chonnam National University Hospital|Institute of Bioequivalence and Bridging Study College of Pharmacy CNU
 March 2008 Not Applicable

Chemical Information & Solubility

Molecular Weight 370.79 Formula

C19H15ClN2O4
CAS No. 90098-04-7 SDF Download Rebamipide SDF
Smiles C1=CC=C2C(=C1)C(=CC(=O)N2)CC(C(=O)O)NC(=O)C3=CC=C(C=C3)Cl
Storage (From the date of receipt)

In vitro
Batch:

DMSO : 74 mg/mL ( (199.57 mM)； Moisture-absorbing DMSO reduces solubility. Please use fresh DMSO.)

Water : Insoluble

Ethanol : Insoluble


Molecular Weight Calculator

In vivo
Batch:

Add solvents to the product individually and in order.


In vivo Formulation Calculator

Preparing Stock Solutions

Molarity Calculator

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In vivo Formulation Calculator (Clear solution)

Step 1: Enter information below (Recommended: An additional animal making an allowance for loss during the experiment)

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Step 2: Enter the in vivo formulation (This is only the calculator, not formulation. Please contact us first if there is no in vivo formulation at the solubility Section.)

% DMSO % % Tween 80 % ddH2O
%DMSO %

Calculation results:

Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO ( Master liquid concentration mg/mL, Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug. )

Method for preparing in vivo formulation: Take μL DMSO master liquid, next addμL PEG300, mix and clarify, next addμL Tween 80, mix and clarify, next add μL ddH2O, mix and clarify.

Method for preparing in vivo formulation: Take μL DMSO master liquid, next add μL Corn oil, mix and clarify.

Note: 1. Please make sure the liquid is clear before adding the next solvent.
2. Be sure to add the solvent(s) in order. You must ensure that the solution obtained, in the previous addition, is a clear solution before proceeding to add the next solvent. Physical methods such
as vortex, ultrasound or hot water bath can be used to aid dissolving.

Tech Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store inhibitors, and issues that need special attention for cell-based assays and animal experiments.

Handling Instructions

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