Prasugrel (Effient) Chemical Structure
GW 791343 hydrochloride is a non-competitive human P2X(7) receptor inhibitor with pIC50 of about 7.1.
LY404039 is a potent agonist of recombinant human mGlu2, mGlu3 receptors and rat neurons expressing native mGlu2/3 receptors with Ki of 149 nM, 92 nM and 88nM, respectively.
COX-2 inhibitor,IC50=0.04uM
BMS-708163 is a γ-secretase inhibitor (GSI) (IC50 =0.3 nM)
Asenapine is a new atypical antipsychotic used for the treatment of schizophrenia and acute mania associated with bipolar disorder .
Cetirizine Dihydrochloride is an antihistamine.
Etodolac (Lodine) is a COX inhibitor with an IC50 of 53.5 nM.
Etomidate is a GABAA receptors agonist at GABAA receptors.
Flumazenil is a benzodiazepine antagonist.
Fluoxetine is an antidepressant of the selective serotonin reuptake inhibitor (SSRI)class.
Prasugrel is a novel platelet inhibitor used for the reduction of thrombotic cardiovascular events (including stent thrombosis) in patients with acute coronary syndrome who are to be managed with PCI. [1]
Prasugrel reduces the aggregation ("clumping") of platelets by irreversibly binding to P2Y12 receptors. In rat platelets, prasugrel AM inhibited in vitro platelet aggregation induced by ADP (10 μm) with an IC50 value of 1.8 μm. [2]
| Molecular Weight (WM): | 373.44 |
|---|---|
| Formula: | C20H20FNO3S |
| CAS No.: | 150322-43-3 |
| Synonyms: |
Effient, Efient, Prasita
|
| Dissolve in (25°C): | DMSO ≥30mg/mL |
| Water <1mg/mL | |
| Ethanol ≥7mg/mL | |
| Storage: | 2 years-20°CPowder |
| 1 week-4°Cin DMSO | |
| 1 month-80°in DMSO |
A collection of 864 bioactive compounds
A collection of 481 inhibitors
A collection of 194 kinase inhibitors
A collection of 85 tyrosine kinase inhibitors.
A collection of 426 FDA approved drugs
A collection of 139 natural products
A collection of 40 chemotherapeutic agents
A unique collection of 17 small molecule modulators
A unique collection of 47 small molecule inhibitors
A unique collection of 63 GPCR small molecules
Keywords:buy Prasugrel (Effient) | Prasugrel (Effient) supplier | purchase Prasugrel (Effient) | Prasugrel (Effient) cost | Prasugrel (Effient) manufacturer | order Prasugrel (Effient) | Prasugrel (Effient) distributor