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S1979
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Amiodarone HCl |
Amiodarone HCl is an antiarrhythmic drug for inhibition of ATP-sensitive potassium channel with IC50 of 19.1 μM.
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S1160
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TRAM-34 |
TRAM-34 is a selective and potent inhibitor of the intermediate-conductance Ca2+-activated K+ channel (IKCa1, KCa3.1) with Kd of 20 nM. |
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S1426
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Repaglinide |
Repaglinide is for the treatment of type II diabetes. |
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S1971
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Nicorandil(Ikorel) |
Nicorandil(Ikorel) is potassium channel activator. |
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S2489
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Nateglinide (Starlix) |
Nateglinide(Starlix) is an insulin secretagog agent that lowers blood glucose levels by stimulating insulin secretion from the pancreas. |
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S2456
|
Chlorpromazine (Sonazine) |
Chlorpromazine (Sonazine) is a dopamine and potassium channel inhibitor with IC50 of 6.1 and 16 μM for nward-rectifying K+ currents and time-independent outward currents |
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S2601
|
Gliclazide (Diamicron) |
Gliclazide (Diamicron) is a whole-cell beta-cell ATP-sensitive potassium currents blocker with an IC50 of 184 ± 30 nM. |
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S8016
|
TAK-438 |
TAK-438 is a novel potassium-competitive acid blocker (P-CAB) type antisecretory agent that reversibly inhibits gastric H+, K+-ATPase with IC50 of 19 nM at pH 6.5. |
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S2443
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Tolbutamide |
Tolbutamide is an inhibitor of cAMP with IC50 of 4 mM. |
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S2073
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Mitiglinide calcium |
Mitiglinide is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-cells.
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S3151
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Gliquidone |
Gliquidone is an ATP-sensitive K+ channel antagonist with IC50 of 27.2 nM. |
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S2825
|
ML133 HCl |
ML133 is a potent potassium channel inhibitor for Kir2.1 with IC50 of 1.8 μM (pH 7.4) and 290 nM (pH 8.5). |
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