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S2882
|
IKK-16 |
IKK 16 is a selective IκB kinase (IKK) inhibitor for IKK-2, IKK complex and IKK-1 with IC50 of 40 nM, 70 nM and 200 nM, respectively. |
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S2824
|
TPCA-1 |
TPCA-1 is an inhibitor of IKK-2 with IC50 of 17.9 nM. |
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S2864
|
IMD 0354 |
IMD-0354 is an IKKβ inhibitor and blocks IκBα phosphorylation in NFκβ pathway. |
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S2913
|
BAY 11-7082 (BAY 11-7821) |
Bay 11-7082 inhibits TNFα-induced IκBα phosphorylation with IC50 of 10 μM. |
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S1274
|
BX-795 |
BX795 is a potent and specific TBK1, IKKε and PDK-1 inhibitor with IC50 of 6 nM, 41 nM and 111 nM, respectively. |
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S4905
|
PHA-408 |
PHA-408 is a highly selective and ATP-competitive IKK-2 inhibitor with IC50 of 40 nM. |
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S4906
|
PF-184 |
PF-184 is a potent and selective IKK-2 inhibitor with IC50 of 37 nM. |
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S4907
|
SC-514 |
SC-514 is an orally active, ATP-competitive IKK-2 inhibitor with IC50 of 3-12 μM. |
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