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Adrenergic Receptor Antagonists & Agonists

Adrenergic Receptor Antagonists & Agonists (48)
water-soluble

Cat.No.	Product Name	Information	Product Citations
S2840	ARN-509	ARN-509 is a selective androgen receptor inhibitor with IC50 of 16 nM.
S1324	Doxazosin mesylate	Doxazosin mesylate is an alpha-1 adrenergic receptor blocker.
S1549	Nebivolol (Bystolic)	Nebivolol selectively inhibits β1-adrenoceptor with IC50 of 0.8 nM.
S1206	Bisoprolol	Bisoprolol is a selective type β1 adrenergic receptor blocker
S1387	Naftopidil DiHCl	Naftopidil DiHCl is a selective 5-HT_1A and α₁-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
S4043	Tetrahydrozoline HCl	Tetrahydrozoline HCl is an imidazoline derivative with alpha receptor agonist activity.
S4009	Mirabegron (YM178)	Mirabegron is a selective β3-adrenoceptor agonist with EC50 of 22.4 nM.
S4010	Acebutolol HCl	Acebutolol is a β-adrenergic receptors antagonist used in the treatment of hypertension, angina pectoris and cardiac arrhythmias.
S1283	Asenapine	Asenapine ihibits adrenergic receptor (α₁, α_2A, α_2B, α_2C) with K_i of 0.25-1.2 nM and also inhibits 5-HT receptor (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) with K_i of 0.03-4.0 nM.
S2521	Epinephrine bitartrate (Adrenalinium)	Epinephrine bitartrate (D02149, Adrenalinium) is alpha- and beta-adrenergic receptor stimulator.
S3061	Epinephrine HCl (Adrenaline)	Epinephrine HCl is a hormone and a neurotransmitter.
S3075	Dexmedetomidine	Dexmedetomidine is a sedative medication used by intensive care units and anesthetists.
S2438	Synephrine HCl	Synephrine HCl (Oxedrine, p-Synephrine) is a sympathomimetic α-adrenergic receptor (AR) agonist.
S2113	Cisatracurium besylate (Nimbex)	Cisatracurium besylate is a nondepolarizing neuromuscular blocking agent, antagonizing the action of acetylcholine by inhibiting neuromuscular transmission.
S2083	Procaterol HCl	Procaterol is a short-acting β2-adrenergic receptor agonist with K_p of 8 nM, used for the treatment of asthma
S2086	Ivabradine HCl (Procoralan)	Ivabradine, a new I_f inhibitor with IC 50 of 2.9 μM which acts specifically on the pacemaker activity of the sinoatrial node, is a pure heart rate lowering agent.
S2090	Dexmedetomidine HCl (Precedex)	Dexmedetomidine is a highly selective and potent alpha-2 adrenoceptor agonist, which reduces anesthetic requirements for patients by providing significant sedation.
S2091	Betaxolol (Betoptic)	Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
S2092	Detomidine HCl	Detomidine produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
S2059	Terazosin HCl (Hytrin)	Hytrin (terazosin) is an alpha-adrenergic blocker used to treat high blood pressure and enlarged prostate.
S1856	Metoprolol tartrate	Metoprolol tartrate is a cardioselective β-adrenergic receptor blocker with IC50 of 42 ng/mL.
S2523	DL-Adrenaline	DL-Adrenaline is a hormone and a neurotransmitter secreted by the medulla of the adrenal glands.
S2545	Scopine	Scopine is the metabolite of anisodine, which is a α1-adrenergic receptor agonist and used in the treatment of acute circulatory shock.
S2038	Phentolamine mesilate	Phentolamine mesilate is a nonselective alpha-adrenergic antagonist with IC50 of 0.1 μM.
S1827	Betaxolol HCl (Betoptic)	Betaxolol hydrochloride (Betoptic) is a β₁ adrenergic receptor blocker with IC50 of 6 μM.
S2020	Formoterol hemifumarate	Formoterol hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist to β2 and β1 receptors with pKd of 8.12 and 5.58, respectively.
S3083	Indacaterol Maleate	Indacaterol is an ultra-long-acting β-adrenoceptor agonist with pK_i of 7.36.
S3060	Medetomidine HCl
S3185	Adrenalone HCl	Adrenalone is an adrenergic agonist.
S3153	Levalbuterol HCl	Levalbuterol HCl is a relatively selective beta2-adrenergic receptor agonist used for the treatment of asthma.
S1831	Carvedilol	Carvedilol is a non-selective beta blocker/alpha-1 blocker with an IC50 of 3.8 μM for inhibition of LDL oxidation.
S2569	Phenylephrine HCl	Phenylephrine hydrochloride is a selective α1-adrenergic receptor agonist.
S2566	Isoprenaline HCl	Isoprenaline is a non-selective β-adrenoceptor, inhibits the ³H-inositol phosphate accumulation with IC50 of 0.08 μM.
S2533	Ritodrine HCl (Yutopar)	Ritodrine hydrochloride (DU 21220; Miolene; NSC 291565; Pre-Par) is a hydrochloride salt of ritodrine which is a β-2 adrenergic receptor agonist.
S2517	Maprotiline HCl	Maprotiline hydrochloride (Deprilept, Ludiomil, Psymion) is a selective noradrenalin re-uptake inhibitor and a tetracyclic antidepressant.
S2519	Naphazoline HCl (Naphcon)	Naphazoline hydrochloride (Naphcon) is an ocular vasoconstrictor and imidazoline derivative sympathomimetic amine.
S2522	L-Adrenaline (Epinephrine)	L-Adrenaline (Epinephrine) belongs to a group of the compounds known as catecholamines.
S2507	Salbutamol sulfate (Albuterol)	Salbutamol (Albuterol) is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 µM.
S2509	Sotalol (Betapace)	Sotalol (Betapace) is a non-selective beta blocker and a potassium channel blocker with an IC50 of 43 μM
S2516	Xylazine HCl	Xylazine HCl is α2 class of adrenergic receptor agonist.	Acad Radiol, 2012, 19(3):358-65
S2458	Clonidine HCl (Catapres)	Clonidine hydrochloride(Catapres) is a direct-acting α2 adrenergic agonist with an ED50 of 0.02±0.01 mg/kg.
S2495	Oxymetazoline HCl	Oxymetazoline hydrochloride is an α1 and α2 adrenergic receptor agonist.
S2499	Phenoxybenzamine HCl	Phenoxybenzamine HCl is a non-specific, irreversible alpha antagonist with an IC50 of 550 nM.
S2126	Naftopidil (Flivas)	Naftopidil (Flivas) is a selective α1-adrenergic receptor antagonist or alpha blocker with a Ki of 58.3 nM.
S1613	Silodosin (Rapaflo)	Silodosin(Rapaflo) is an α1-adrenoceptor antagonist with high uroselectivity.
S1427	Rilmenidine	Rilmenidine is a second-generation imidazoline-α2 adrenergic agonist.
S1437	Tizanidine HCl	Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
S1409	Alfuzosin HCl(Uroxatral)	Alfuzosin(Uroxatral) is an alpha1 receptor antagonist used to treat benign prostatic hyperplasia (BPH).

Inhibitory Selectivity
Solubility

Cat.No.	Product Name	Solubility (25°C)
Cat.No.	Product Name	Water	DMSO	Ethanol
S2840	ARN-509	<1 mg/mL	18 mg/mL	5 mg/mL
S1324	Doxazosin mesylate	<1 mg/mL	15 mg/mL	<1 mg/mL
S1549	Nebivolol (Bystolic)	<1 mg/mL	88 mg/mL	<1 mg/mL
S1206	Bisoprolol	88 mg/mL	88 mg/mL	88 mg/mL
S1387	Naftopidil DiHCl	<1 mg/mL	41 mg/mL	2 mg/mL
S4043	Tetrahydrozoline HCl	47 mg/mL	12 mg/mL	26 mg/mL
S4009	Mirabegron (YM178)	<1 mg/mL	79 mg/mL	8 mg/mL
S4010	Acebutolol HCl	75 mg/mL	75 mg/mL	75 mg/mL
S1283	Asenapine	<1 mg/mL	80 mg/mL	<1 mg/mL
S2521	Epinephrine bitartrate (Adrenalinium)	67 mg/mL	67 mg/mL	<1 mg/mL
S3075	Dexmedetomidine	40 mg/mL	40 mg/mL	40 mg/mL
S2438	Synephrine HCl	41 mg/mL	14 mg/mL	4 mg/mL
S2113	Cisatracurium besylate (Nimbex)	47 mg/mL	249 mg/mL	249 mg/mL
S2086	Ivabradine HCl (Procoralan)	82 mg/mL	101 mg/mL	101 mg/mL
S2090	Dexmedetomidine HCl (Precedex)	<1 mg/mL	48 mg/mL	48 mg/mL
S2091	Betaxolol (Betoptic)	62 mg/mL	62 mg/mL	<1 mg/mL
S2092	Detomidine HCl	45 mg/mL	45 mg/mL	45 mg/mL
S2059	Terazosin HCl (Hytrin)	<1 mg/mL	26 mg/mL	<1 mg/mL
S2523	DL-Adrenaline	<1 mg/mL	0.02 mg/mL	<1 mg/mL
S2545	Scopine	31 mg/mL	31 mg/mL	31 mg/mL
S2038	Phentolamine mesilate	76 mg/mL	76 mg/mL	76 mg/mL
S1827	Betaxolol HCl (Betoptic)	69 mg/mL	69 mg/mL	69 mg/mL
S2020	Formoterol hemifumarate	<1 mg/mL	98 mg/mL	<1 mg/mL
S3083	Indacaterol Maleate	<1 mg/mL	102 mg/mL	<1 mg/mL
S3060	Medetomidine HCl	47 mg/mL	12 mg/mL	47 mg/mL
S3185	Adrenalone HCl	44 mg/mL	44 mg/mL	<1 mg/mL
S1831	Carvedilol	<1 mg/mL	81 mg/mL	4 mg/mL
S2569	Phenylephrine HCl	41 mg/mL	41 mg/mL	41 mg/mL
S2566	Isoprenaline HCl	50 mg/mL	50 mg/mL	<1 mg/mL
S2533	Ritodrine HCl (Yutopar)	65 mg/mL	65 mg/mL	65 mg/mL
S2517	Maprotiline HCl	<1 mg/mL	63 mg/mL	24 mg/mL
S2519	Naphazoline HCl (Naphcon)	49 mg/mL	17 mg/mL	22 mg/mL
S2522	L-Adrenaline (Epinephrine)	<1 mg/mL	4 mg/mL	<1 mg/mL
S2507	Salbutamol sulfate (Albuterol)	68 mg/mL	<1 mg/mL	<1 mg/mL
S2509	Sotalol (Betapace)	62 mg/mL	62 mg/mL	<1 mg/mL
S2516	Xylazine HCl	12 mg/mL	50 mg/mL	50 mg/mL
S2458	Clonidine HCl (Catapres)	53 mg/mL	53 mg/mL	53 mg/mL
S2495	Oxymetazoline HCl	59 mg/mL	59 mg/mL	59 mg/mL
S2499	Phenoxybenzamine HCl	17 mg/mL	68 mg/mL	68 mg/mL
S2126	Naftopidil (Flivas)	<1 mg/mL	79 mg/mL	<1 mg/mL
S1613	Silodosin (Rapaflo)	<<1 mg/mL	99 mg/mL	99 mg/mL
S1437	Tizanidine HCl	15 mg/mL	10 mg/mL	<1 mg/mL
S1409	Alfuzosin HCl(Uroxatral)	85 mg/mL	85 mg/mL	85 mg/mL

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Adrenergic Receptor Antagonists & Agonists

Adrenergic Receptor Antagonists & Agonists (48)water-soluble

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Adrenergic Receptor Antagonists & Agonists (48)
water-soluble