Research Area
Product Type
PKC Inhibitors
- Cat.No
- Product Name
- Information
- Publications
- Customer Reviews
S5002- Fingolimod (FTY720)
- Fingolimod (FTY720) Gilenia is Src-bcr-Abl Inhibitor & S1P receptor agonist with IC50 of 0.137, 10.98 nM for (S)- and (R)- FTY720-phosphate.
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(1) 
(0)
- S1055
- Enzastaurin (LY317615)
- Enzastaurin (LY317615) is a potent PKC beta inhibitor for PKCβ, PKCα, PKCγ and PKCε with IC50 of 6 nM, 39 nM, 83 nM and 110 nM, respectively.
(0)
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S1314
- Zoledronic Acid (Zoledronate)
- A potent nitrogen-containing bisphosphonates.It inhibited proliferation of human foetal osteoblastic cell line (hFOB) with an IC50 of 40 μM.
- (0)
- (0)
- S2248
- CX-4945
- CX-4945 is a potent and selective ATP-competitive small molecule protein kinase CK2 inhibitor with a Ki and an IC50 of 0.38 and 1 nM for recombinant human CK2α, respectively.
- (0)
- (0)
- S2391
- Quercetin (Sophoretin)
- Quercetin (Sophoretin) is a PI3K and PKC inhibitor with IC50 of 3.8 μM and 15µg/ml.
- (0)
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(1)
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S1292
- Chelerythrine Chloride
- Chelerythrine is a potent, selective, and cell-permeable PKC inhibitor (IC50 = 660 nM).
- (0)
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