PPAR Inhibitors

Cat.No.	Product Name	Information
S2505	Rosiglitazone maleate	Rosiglitazone maleate (Avandia) is an anti-diabetic agent in the thiazolidinedione class of agents.
S2915	GW9662	GW9662 is a selective PPAR antagonist, inhibiting PPARγ, PPARα and PPARδ with IC50 of 3.3 nM, 32 nM and 2 μM, respectively.
S2556	Rosiglitazone (Avandia)	Rosiglitazone (Avandia) is a potent antihyperglycemic agent and a potent thiazolidinedione insulin sensitizer with IC50 of 12, 4 and 9 nM for rat, 3T3-L1 and human adipocytes, respectively.
S2871	T0070907	T0070907 is a potent and selective PPARγ inhibitor with IC50 of 1 nM.
S1473	GW501516	GW501516 is a selective PPARδ agonist with K_i of 1.1 nM.
S8029	WY 14643 (Pirinixic Acid)	WY 14643 (Pirinixic Acid) is a potent peroxisome proliferator and activator of PPAR alpha.
S8026	GSK0660	GSK0660 is a selective PPARδ antagonist with IC50 of 155 nM.
S8046	GW7647	GW7647 is a potent and highly selective PPARα agonist with EC50 of 6 nM.
S8020	GW0742	GW0742 is a potent and highly selective PPARβ/δ agonist, binding to hPPARδ with IC50 of 1 nM.
S2665	Ciprofibrate	Ciprofibrate is a peroxisome proliferator-activated receptor agonist.
S2075	Rosiglitazone HCl	Rosiglitazone is a blood glucose-lowering drugs, stimulating insulin secretion by binding to the PPAR receptors in fat cells.
S2798	GW6471	GW6471 is an inhibitor of PPARα with IC50 of 0.24 μM.

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