PDK-1 Inhibitors

Cat.No.	Product Name	Information	Product Citations
S1275	BX-912	BX912 is a selective potent PDK1 inhibitor with IC50 of 12 nM.
S1274	BX-795	BX795 is a potent and specific TBK1, IKKε and PDK-1 inhibitor with IC50 of 6 nM, 41 nM and 111 nM, respectively.
S1106	OSU-03012	OSU-03012 is a potent inhibitor of recombinant PDK-1 with IC50 of 5 μM.	Am J Physiol Renal Physiol, 2011, 302(4), F466-76 Eukaryot Cell, 2012, 12(1), 12-22
S1556	PHT-427	PHT-427 is a dual Akt and PDPK1 inhibitor with K_i of 2.7 μM and 5.2 μM, respectively.	Blood, 2011, 118(10), 2840-2848

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