Other Inhibitors

• Cat.No
• Product Name
• Information
• Publications
• Customer Reviews

• S6003
• PTC124 (Ataluren)
• PTC124 also known as Ataluren is CFTR-G542X nonsense allele inhibitor.
• (1)
• (1)

• S1453
• Tipifarnib (Zarnestra)
• Tipifarnib (Zarnestra) is a potent and specific farnesyltransferase inhibitor with an IC50 of 0.6 nM.
• (0)
• (0)

• S1565
• VX-809
• VX-809 is the second investigational oral candidate compound for the treatment of cystic fibrosis (CF).
• (0)
• (0)

• S5003
• FK-506 (Tacrolimus)
• An immunosuppressive agent and macrolide antibiotic.
• (0)
• (0)

• S1113
• GSK690693
• GSK690693 is a pan-Akt kinase inhibitor,IC50 of Akt 1, 2, and 3 at 2, 13, and 9 nM respectively.
• (0)
• (0)

• S1257
• Posaconazole
• Posaconazole is a triazole antifungal agent.
• (0)
• (0)

• S1237
• Methazolastone
• P.o. imidazotetrazine second-generation alkylating agent.
• (0)
• (0)

• S1162
• PA-824
• PA-824 is an experimental anti-tuberculosis drug with MIC of less than 1 μg/mL for tuberculosis.
• (0)
• (0)

• S2748
• Anacetrapib (MK-0859)
• Anacetrapib is a potent and selective rhCETP and C13S CETP mutant inhibitor with IC50 of 7.9 nM and 11.8 nM, respectively
• (0)
• (0)

• S2754
• AT-406
• AT-406 is a potent and orally bioavailable IAP (inhibitor of apoptosis protein) inhibitor of XIAP, cIAP1, and cIAP2 proteins with K_i of 66.4, 1.9, and 5.1 nM, respectively.
• (0)
• (0)

• S2666
• PF-3845
• PF-3845 is a potent, selective, and irreversible fatty acid amide hydrolase (FAAH) inhibitor with a Ki of 0.23 μM.
• (0)
• (0)

• S2612
• Ribitol (Adonitol)
• Ribitol (Adonitol) is a sugar alcohol formed by the reduction of ribose.
• (0)
• (0)

• S2416
• Chondroitin sulfate
• Chondroitin sulfate is a kind of sulfated glycosaminoglycan (GAG) which is composed of a chain of alternating sugars including N-acetylgalactosamine and glucuronic acid.
• (0)
• (0)

• S2694
• WAY-362450
• WAY-362450 is a highly potent, selective, and orally active farnesoid X receptor (FXR) agonist with an EC50 of 4 nM.
• (0)
• (0)

• S2155
• LY2608204
• LY2608204 is a potent agent used to treat type 2 diabetes.
• (0)
• (0)

• S2632
• BMS-806 (BMS 378806)
• BMS-806 (BMS 378806) is a small molecule gp120/CD4 inhibitor with an IC50 of median 5 nM.
• (0)
• (0)

• S2156
• LY2886721
• LY2886721 is a novel potent agent that is used to treat Alzheimer's Disease in preclinical experiments.
• (0)
• (0)

• S2526
• Alizarin
• Alizarin is an organic compound and an important prominent dye.
• (0)
• (0)

• S2332
• Neohesperidin
• Neohesperidin is an antioxidant agent with an IC50 of 22.31 μg/ml in the 1,1-diphenyl-2-picryldydrazyl (DPPH) radical-scavenging assay.
• (0)
• (0)

• S2532
• L-Ascorbyl 6-palmitate
• L-Ascorbyl 6-palmitate is a synthetic lipophilic ascorbic acid derivative.
• (0)
• (0)

• S2530
• 7-Aminocephalosporanic acid
• 7-Aminocephalosporanic acid is a key intermediate required for the production of most of the clinically used cephalosporin derivatives.
• (0)
• (0)

• S2404
• Isoliquiritigenin
• Isoliquiritigenin (GU 17) is a strong nod gene- and glyceollin resistance-inducing flavonoid from soybean root exudate.
• (0)
• (0)

• S2405
• Sophocarpine
• Sophocarpine is a human ether-à-go-go-related gene (HERG) inhibitor with an IC(50) of about 0.2 mM.
• (0)
• (0)

• S2407
• Curcumol
• Curcumol is a common traditional Chinese medicine with antitumor activities.
• (0)
• (0)

• S2400
• Rhein(Monorhein)
• Rhein(Monorhein; NSC 38629; Rheic acid; Rheinic acid) is a constituent of rhubarb which was isolated from the fresh rhizome of Rheum coreanum Nakai.
• (0)
• (0)

• S2402
• Cyclovirobuxin D(Bebuxine)
• Cyclovirobuxine D (bebuxine; Cyclovirobuxine) is an active compound extracted from Buxus microphylla, which has been used for treating acute myocardial ischemia.
• (0)
• (0)

• S2395
• Rheochrysidin (Physcione)
• Rheochrysidin (Physcion; physcione; parietin) is one of the major components of Da-Cheng-Qi decoction used in the treatment of inflammation.
• (0)
• (0)

• S2396
• Salidroside(Rhodioloside)
• Salidroside (Rhodioloside; Rhodosin) is a glucoside compound with an IC50 of 4.99 ± 0.23 μg/mL for the proliferation of SACC-2 cells.
• (0)
• (0)

• S2397
• Palmatine chloride
• Palmatine hydrochloride (Palmatine chloride (6CI,7CI); Fibrauretin) is a hydrochloride salt of palmatine which is a protoberberine alkaloid.
• (0)
• (0)

• S2398
• Coenzyme Q10 (CoQ10)
• Coenzyme Q10 (ubiquinone, ubidecarenone, coenzyme Q) is a component of the electron transport chain and participates in aerobic cellular respiration.
• (0)
• (0)

• S2399
• Dihydromyricetin(Ampeloptin)
• Dihydromyricetin (Ampelopsin, flavanol, Ampeloptin) is a natural antioxidant with good prospects.
• (0)
• (0)

• S2385
• Hordenine
• Hordenine (N,N-dimethyl-4-hydroxyphenylethylamine) is a phenylethylamine alkaloid with antibacterial and antibiotic properties.
• (0)
• (0)

• S2382
• Evodiamine (Isoevodiamine)
• Evodiamine (Isoevodiamine) is an alkaloid extract from a plant known as Evodiae Fructus.
• (0)
• (0)

• S2383
• Gastrodin (Gastrodine)
• Gastrodin (Gastrodine) is a polyphenol. It is the glucoside of 4-hydroxybenzyl alcohol (gastrodigenin).
• (0)
• (0)

• S2384
• Hematoxylin (Hydroxybrazilin)
• Hematoxylin (Hydroxybrazilin) is a compound that forms strongly colored complexes with certain metal ions, notably Fe(III) and Al(III) salts and a kind of stain in histology.
• (0)
• (0)

• S2387
• Lappaconite Hydrobromide
• Lappaconite Hydrobromide is a kind of alkaloid extracted from Aconitum sinomontanum Nakai and has anti-inflammatory effects.
• (0)
• (0)

• S2389
• Naringin Dihydrochalcone(Naringin DC)
• Naringin Dihydrochalcone(Naringin DC) is a new-style sweetening agent and an artificial sweetener derived from naringin.
• (0)
• (0)

• S2390
• Polydatin(Piceid)
• Polydatin(Piceid), 3,4’,5-trihydroxystilbene-3-β-mono-D-glucoside, the crystal component extracted from the root stem of perennial herbage Polygonum Cuspidatum Sieb.et Zucc.
• (0)
• (0)

• S2392
• Sesamin(Fagarol)
• Sesamin(Fagarol) is a lignan isolated from the bark of Fagara plants and from sesame oil.
• (0)
• (0)

• S2374
• 5-hydroxytryptophan (5-HTP)
• 5-Hydroxytryptophan(5-HTP) is decarboxylated to serotonin (5-hydroxytryptamine or 5-HT) by the enzyme aromatic-L-amino-acid decarboxylase with the help of Vitamin B6.
• (0)
• (0)

• S2375
• Aloin (Barbaloin)
• Aloin(Barbaloin) is a potent tyrosinase inhibitor with an IC50 of 97 μM for HeLaS3 cells
• (0)
• (0)

• S2377
• Biochanin A (4-Methylgenistein)
• Biochanin A(4-Methylgenistein) is an O-methylated isoflavone. It is a natural organic compound in the class of phytochemicals known as flavonoids.
• (0)
• (0)

• S2379
• Dioscin (Collettiside III)
• Dioscin(Collettiside III) is a saponin extracted and isolated from Polygonatum Zanlanscianense Pamp with IC50 of 2.6, 0.8, 7.5, and 4.5 μM for the inhibition of the growth of the MDA-MB-435, H14, HL60, and HeLa cell lines, respectively.
• (0)
• (0)

• S2380
• Diosmetin(Luteolin 4-methyl ether)
• Diosmetin (Luteolin 4-methyl ether) is a bioflavonoid found in spearmint, oregano, and many other plants.
• (0)
• (0)

• S2457
• Clindamycin hydrochloride (Dalacin)
• Clindamycin hydrochloride(Dalacin) is the hydrated hydrochloride salt of clindamycin which is a semisynthetic antibiotic.
• (0)
• (0)

• S2371
• Vanillylacetone
• Vanillylacetone is similar in chemical structure to other flavor chemicals such as vanillin and eugenol. It is used as a flavor additive in spice oils and in perfumery to introduce spicy aromas.
• (0)
• (0)

• S2372
• Xanthone (Genicide)
• Xanthone is an organic compound. It can be prepared by the heating of phenyl salicylate.
• (0)
• (0)

• S2373
• Yohimbine hydrochloride (Antagonil)
• Yohimbine(Antagonil) has been used as a mydriatic and in the treatment of impotence. It is also alleged to be an aphrodisiac.
• (0)
• (0)

• S2352
• Salinomycin (Procoxacin)
• Salinomycin (Procoxacin) is an antibacterial and coccidiostat ionophore therapeutic agent.
• (0)
• (0)

• S2354
• Sclareol
• Sclareol is a fragrant chemical compound found in clary sage (Salvia sclarea), from which it derives its name. It is classified as a bicyclic diterpene alcohol.
• (0)
• (0)

• S2355
• Sclareolide (Norambreinolide)
• Sclareolide(Norambreinolide) is a sesquiterpene lactone natural product derived from various plant sources including Salvia sclarea, Salvia yosgadensis, and cigar tobacco.
• (0)
• (0)

• S2356
• Shikimic acid (Shikimate)
• Shikimic acid(Shikimate), more commonly known as its anionic form shikimate, is an important biochemical intermediate in plants and microorganisms.
• (0)
• (0)

• S2357
• Silibinin (Silybin)
• Silibinin(Silybin) is the major active constituent of silymarin.
• (0)
• (0)

• S2358
• Silymarin (Silybin B)
• Silymarin(Silybin B), a strong novel free radical scavenger, is used for treatment of patients with acute brain infarction.
• (0)
• (0)

• S2359
• Sinomenine (Cucoline)
• Sinomenine(Cucoline) is traditionally used in herbal medicine in these countries, as a treatment for rheumatism and arthritis.
• (0)
• (0)

• S2361
• Stigmasterol (Stigmasterin)
• Stigmasterol(Stigmasterin) is used as a precursor in the manufacture of synthetic progesterone.
• (0)
• (0)

• S2363
• Tangeretin (Tangeritin)
• Tangeretin(Tangeritin) is a citrus flavonoids.
• (0)
• (0)

• S2364
• Tanshinone I
• Tanshinone I is isolated from Danshen.
• (0)
• (0)

• S2365
• Tanshinone IIA (Tanshinone B)
• Tanshinone IIA(Tanshinone B) is the most abundant diterpene quinone in Danshen, Salviae miltiorrhizae Radix, a widely prescribed traditional herbal medicine that is used to treat cardiovascular and inflammatory diseases.
• (0)
• (0)

• S2366
• Taxifolin (Dihydroquercetin)
• Taxifolin(Dihydroquercetin) is a flavanonol, a type of flavonoid.
• (0)
• (0)

• S2367
• Tetrahydropapaverine hydrochloride
• Tetrahydropapaverine, one of the TIQs and an analogue of salsolinol and tetrahydropapaveroline, has been reported to have neurotoxic effects on dopamine neurons.
• (0)
• (0)

• S2368
• Theobromine (3,7-Dimethylxanthine)
• Theobromine(3,7-Dimethylxanthine) is a xanthine alkaloid that is used as a bronchodilator and as a vasodilator.
• (0)
• (0)

• S2369
• Troxerutin
• Troxerutin(Trihydroxyethylrutin) is a flavonol, a type of flavonoid.
• (0)
• (0)

• S2370
• Ursolic acid (Malol)
• Ursolic acid(Malol) is a pentacyclic triterpene acid, used in cosmetics.
• (0)
• (0)

• S2341
• Parthenolide ((-)-Parthenolide)
• Parthenolide ((-)-Parthenolide) is a sesquiterpene lactone which occurs naturally in the plant feverfew (Tanacetum parthenium).
• (0)
• (0)

• S2342
• Phloretin (Dihydronaringenin)
• Phloretin(Dihydronaringenin) is a dihydrochalcone, a type of polyphenol.
• (0)
• (0)

• S2343
• Phlorizin (Phloridzin)
• Phlorizin (Phloridzin) is a toxic 2’-glucoside of phloretin. It belongs to the group of dihydrochalcones, a type of flavonoids.
• (0)
• (0)

• S2344
• Piperine (1-Piperoylpiperidine)
• Piperine(1-Piperoylpiperidine) is the alkaloid responsible for the pungency of black pepper and long pepper, along with chavicine (an isomer of piperine). It has also been used in some forms of traditional medicine and as an insecticide.
• (0)
• (0)

• S2346
• Puerarin (Kakonein)
• Puerarin (Kakonein) is a 5-HT2C receptor and benzodiazepine site antagonist.
• (0)
• (0)

• S2347
• Quercetin dihydrate (Sophoretin)
• Quercetin, a flavonol widely distributed in plants. It is an antioxidant, like many other phenolic heterocyclic compounds.
• (0)
• (0)

• S2349
• Rutaecarpine (Rutecarpine)
• Rutaecarpine is an indolopyridoquinazolinone alkaloid isolated from Evodia rutaecarpa and related herbs.
• (0)
• (0)

• S2350
• Rutin (Rutoside)
• Rutin, a flavonol glycoside found in many plants, including buckwheat; tobacco; forsythia; hydrangea; viola, etc.
• (0)
• (0)

• S2351
• Salicin (Salicoside, Salicine)
• Salicin(Salicoside, Salicine) is an alcoholic β-glycoside that contains D-glucose. Salicin is an anti-inflammatory agent that is produced from willow bark.
• (0)
• (0)

• S1893
• D-glutamine
• D-glutamine is one of the 20 amino acids encoded by the standard genetic code.
• (0)
• (0)

• S2324
• Monensin sodium salt (Coban)
• Monensin sodium salt(Coban), isolated from Streptomyces cinnamonensis, is a well-known representative of naturally polyether ionophore antibiotics.
• (0)
• (0)

• S2325
• Morin hydrate (Aurantica)
• Morin hydrate(Aurantica) is a chemical compound. Morin can be used to test for the presence of aluminum or tin in a solution, since it forms characteristically fluorescent coordination complexes with them.
• (0)
• (0)

• S2326
• Myricetin (Cannabiscetin)
• Myricetin(Cannabiscetin) is a naturally occurring flavonol, a flavonoid found in many grapes, berries, fruits, vegetables, herbs, as well as other plants.
• (0)
• (0)

• S2327
• Myricitrin (Myricitrine)
• Myricitrin(Myricitrine) is a chemical compound. It can be isolated from the root bark of Myrica cerifera (Bayberry, a small tree native to North America) and in Chrysobalanus icaco.
• (0)
• (0)

• S2329
• Naringin (Naringoside)
• Naringin (Naringoside) is a flavanone glycoside and is a major flavonoid in grapefruit and gives the grapefruit juice its bitter taste.
• (0)
• (0)

• S2330
• Nattokinase
• Nattokinase is an enzyme extracted and purified from a Japanese food called nattō.
• (0)
• (0)

• S2331
• Neohesperidin dihydrochalcone (Nhdc)
• Neohesperidin dihydrochalcone(Nhdc), sometimes abbreviated to neohesperidin DC or simply NHDC, is an artificial sweetener derived from citrus.
• (0)
• (0)

• S2333
• Nobiletin (Hexamethoxyflavone)
• Nobiletin (Hexamethoxyflavone) is a chemical compound and an O-methylated flavone, a flavonoid isolated from citrus peels like in tangerine.
• (0)
• (0)

• S2334
• Oleanolic Acid (Caryophyllin)
• Oleanolic acid(Caryophyllin) is a naturally occurring triterpenoid, widely distributed in food and medicinal plants, related to betulinic acid. It is relatively non-toxic, antitumor, and hepatoprotective, as well as exhibiting antiviral.properties.
• (0)
• (0)

• S2335
• Oridonin (Isodonol)
• Oridonin(Isodonol), an entkaurane diterpenoid isolated from Rabdosia rubescens, is an important traditional Chinese herbal remedy.
• (0)
• (0)

• S2336
• Orotic acid (6-Carboxyuracil)
• Orotic acid(6-Carboxyuracil) is a heterocyclic compound and an acid.
• (0)
• (0)

• S2337
• Osthole (Osthol)
• Osthole(Osthol) is a type of coumarin.
• (0)
• (0)

• S2338
• Oxymatrine (Matrine N-oxide)
• Oxymatrine(Matrine N-oxide) is one of components of the root of Sophora flavescens.
• (0)
• (0)

• S2339
• Paeonol (Peonol)
• Paeonol(Peonol) is a major component extracted from Chinese herbs moutan cortex and Cynanchum paniculatum .
• (0)
• (0)

• S2316
• Kinetin (6-Furfuryladenine)
• Kinetin(6-Furfuryladenine) is a kind of cytokinin, a class of plant hormone that promotes cell division. Kinetin is often used in plant tissue culture for inducing formation of callus (in conjunction with auxin) and to regenerate shoot tissues from callus.
• (0)
• (0)

• S2317
• L(+)-Rhamnose Monohydrate
• L(+)-Rhamnose (Rham) is a naturally-occurring deoxy sugar.
• (0)
• (0)

• S2319
• Limonin
• Limonin is also known as limonoate D-ring-lactone and limonoic acid di-delta-lactone. Chemically, it is a member of the class of compounds known as furanolactones.
• (0)
• (0)

• S2321
• Magnolol
• Magnolol (2,2'-Bichavicol) is a bioactive compound found in the bark of the Houpu magnolia (Magnolia officinalis).
• (0)
• (0)

• S2322
• Matrine ((+)-Matrine)
• Matrine((+)-Matrine) is an alkaloid found in plants from the Sophora family. It has a variety of pharmacological effects, including anti-cancer effects, and action as a kappa opioid receptor agonist.
• (0)
• (0)

• S2323
• Methyl-Hesperidin
• Methyl-Hesperidin is a flavanone glycoside (flavonoid) (C28H34O15) found abundantly in citrus fruits. Its aglycone form is called hesperetin.
• (0)
• (0)

• S2304
• Gramine
• Gramine is a naturally occurring indole alkaloid present in several plant species.
• (0)
• (0)

• S2306
• Gynostemma Extract
• Gynostemma Extract is a saponins extract derived from the Gynostemma pentaphyllum.
• (0)
• (0)

• S2309
• Hesperidin
• Hesperidin is a flavanone glycoside found abundantly in citrus fruits.
• (0)
• (0)

• S2310
• Honokiol
• Honokiol is a biphenolic compound present in the cones, bark, and leaves of Magnolia grandifloris.
• (0)
• (0)

• S2311
• Hyodeoxycholic acid (HDCA)
• Hyodeoxycholic(HDCA) acid is a secondary bile acid, one of the metabolic byproducts of intestinal bacteria.
• (0)
• (0)

• S2313
• Indole-3-carbinol
• Indole-3-carbinol is produced by the breakdown of the glucosinolate glucobrassicin, which can be found at relatively high levels in cruciferous vegetables.
• (0)
• (0)

• S2314
• Kaempferol
• Kaempferol is a natural flavonol, a type of flavonoid, that has been isolated from plant sources.
• (0)
• (0)

• S1924
• Indocyanine green(Cardiogreen)
• Indocyanine green(Cardiogreen) is a cyanine dye used in medical diagnostics. It is used for determining cardiac output, hepatic function, and liver blood flow, and for ophthalmic angiography.
• (0)
• (0)

• S2271
• Berberine Hydrochloride
• Berberine Hydrochloride is a quaternary ammonium salt from the group of isoquinoline alkaloids.
• (0)
• (0)

• S2273
• β-Sitosterol
• β-Sitosterol is one of several phytosterols (plant sterols) with chemical structures similar to that of cholesterol.
• (0)
• (0)

• S2276
• Bilobalide
• Bilobalide is a biologically active terpenic trilactone present in Ginkgo biloba.
• (0)
• (0)

• S2277
• Caffeic acid
• Caffeic acid is a hydroxycinnamic acid, a naturally occurring organic compound.
• (0)
• (0)

• S2280
• Chlorogenic acid
• Chlorogenic acid is a hydroxycinnamic acid and a member of a family of naturally occurring organic compounds.
• (0)
• (0)

• S2281
• Chrysin
• Chrysin is a naturally occurring flavone chemically extracted from the blue passion flower (Passiflora caerulea).
• (0)
• (0)

• S2282
• Cinchonidine
• Cinchonidine is an alkaloid used in asymmetric synthesis in organic chemistry.
• (0)
• (0)

• S2287
• Cytisine (Baphitoxine, Sophorine)
• Cytisine is a nicotinic acetylcholine receptor agonist.
• (0)
• (0)

• S2289
• Daidzin
• Daidzin is a natural organic compound in the class of phytochemicals known as isoflavones.
• (0)
• (0)

• S2290
• Dihydroartemisinin (DHA)
• Dihydroartemisinin (DHA) is a semi-synthetic derivative of artemisinin and isolated from the traditional Chinese herb Artemisia annua.
• (0)
• (0)

• S2291
• Diosgenin
• Diosgenin is a steroid sapogenin and the precursor for the semisynthesis of progesterone which in turn was used in early combined oral contraceptive pills.
• (0)
• (0)

• S2292
• Diosmin
• Diosmin is a semisynthetic phlebotropic agent and a member of the flavonoid family.
• (0)
• (0)

• S2294
• Ecdysone
• Ecdysone is a steroidal prohormone of the major insect molting hormone 20-hydroxyecdysone, which is secreted from the prothoracic glands.
• (0)
• (0)

• S2295
• Emodin
• Emodin is a purgative resin, 6-methyl-1,3,8-trihydroxyanthraquinone, from rhubarb, the buckthorn and Japanese Knotweed (Fallopia japonica).
• (0)
• (0)

• S2296
• Enoxolone (Glycyrrhetin)
• Enoxolone is a pentacyclic triterpenoid derivative of the beta-amyrin type obtained from the hydrolysis of glycyrrhizic acid, which was obtained from the herb liquorice.
• (0)
• (0)

• S2297
• Ergosterol
• Ergosterol is a sterol and a biological precursor (a provitamin) to vitamin D2.
• (0)
• (0)

• S2298
• Fisetin (Fustel)
• Fisetin (Fustel) is a potent sirtuin activating compound (STAC) and an agent that modulates sirtuins.
• (0)
• (0)

• S2299
• Formononetin (Formononetol)
• Formononetin(Formononetol) is a phytoestrogen from the root of Astragalus membranaceus and an O-methylated isoflavone.
• (0)
• (0)

• S2300
• Fumalic acid (Ferulic acid)
• Fumalic acid(Ferulic acid) is a hydroxycinnamic acid and a type of organic compound found in the Ferula assafoetida L. or Ligusticum chuanxiong.
• (0)
• (0)

• S2301
• Genistin (Genistoside)
• Genistin(Genistoside) is an isoflavone found in a number of dietary plants like soy and kudzu.
• (0)
• (0)

• S2302
• Glycyrrhizic acid
• Glycyrrhizic acid is a widely used anti-inflammatory agent isolated from the licorice root.
• (0)
• (0)

• S2303
• Gossypol
• Gossypol is a polyphenolic aldehyde that permeates cells and acts as an inhibitor for several dehydrogenase enzymes.
• (0)
• (0)

• S2250
• (-)-Epigallocatechin gallate
• (-)-Epigallocatechin gallate is a potent anti-oxidant polyphenol flavonoid isolated from green tea.
• (0)
• (0)

• S2252
• (+)-Usniacin (D-Usnic acid)
• (+)-Usniacin(D-Usnic acid) is a naturally occurring dibenzofuran derivative found in several lichen species.
• (0)
• (0)

• S2253
• 3-Indolebutyric acid (IBA)
• 3-Indolebutyric acid(IBA) is a plant hormone in the auxin family and is an ingredient in many commercial plant rooting horticultural products.
• (0)
• (0)

• S2256
• 4-Methylumbelliferone(4-MU)
• 4-Methylumbelliferone is a hyaluronic acid (HA) synthesis inhibitor with an IC50 of 0.4 mM.
• (0)
• (0)

• S2258
• Aesculin (Esculin)
• Aesculin(Esculin) is a glucoside found in horse chestnuts.
• (0)
• (0)

• S2259
• Aloe-emodin
• Aloe-emodin is an interferon-inducing agent with IC50 of about 1 μg/mL for JEV and of about 0.33 μg/mL for EV71.
• (0)
• (0)

• S2260
• Amygdalin
• Amygdalin is a glycoside initially isolated from the seeds of the tree Prunus dulcis, also known as bitter almonds.
• (0)
• (0)

• S2261
• Andrographolide
• Andrographolide is a labdane diterpenoid that is the main bioactive component of the medicinal plant Andrographis paniculata.
• (0)
• (0)

• S2263
• Arbutin (Uva, p-Arbutin)
• Arbutin(Uvasol, p-Arbutin) is a tyrosinase inhibitor with an IC50 of 1.09 mM.
• (0)
• (0)

• S2265
• Artesunate
• Artesunate is a part of the artemisinin group of agents with an IC50 of < 5 μM for small cell lung carcinoma cell line H69.
• (0)
• (0)

• S2267
• Azomycin (2-Nitroimidazole)
• Azomycin(2-Nitroimidazole) is an antimicrobial antibiotic produced by a strain of Nocardia mesenterica.
• (0)
• (0)

• S2269
• Baicalin
• Baicalin is a known prolyl endopeptidase inhibitor and affects the GABA receptors.
• (0)
• (0)

• S2270
• Bergenin (Cuscutin)
• Bergenin (Cuscutin) is trihydroxybenzoic acid glycoside and the C-glycoside of 4-O-methyl gallic acid.
• (0)
• (0)

• S2000
• Sodium orthovanadate
• Sodium orthovanadate is the chemical compound Na3VO4 and contains the tetrahedral VO43. It is an inhibitor of protein tyrosine phosphatases, alkaline phosphatases and a number of ATPases, most likely acting as a phosphate analogue.
• (0)
• (0)

• S2008
• Taurine
• Taurine, or 2-aminoethanesulfonic acid, is an organic acid.
• (0)
• (0)

• S1655
• Ezetimibe (Zetia)
• Ezetimibe (Zetia) is a compound that lowers cholesterol.
• (0)
• (0)

• S1950
• Metformin hydrochloride(Glucophage)
• Metformin hydrochloride(Glucophage) is a biguanide hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietary modification.
• (0)
• (0)

• S1760
• Rifapentine (Priftin)
• Rifapentine (Priftin) is an antibiotic compound used in the treatment of tuberculosis.
• (0)
• (0)

• S1751
• Gadodiamide (Omniscan)
• Gadodiamide(Omniscan) is a gadolinium-based contrast agent used in MR imaging procedures to assist in the visualization of blood vessels.
• (0)
• (0)

• S2485
• Mitoxantrone Hydrochloride
• Mitoxantrone Hydrochloride (NSC301739, Immunex) is a hydrochloride salt of mitoxantrone which is a synthetic antineoplastic anthracenedione (IC50 = 0.42 mM).
• (0)
• (0)

• S1545
• SB-408124
• SB-408124 is a non-peptide antagonist selective for the orexin receptor subtype OX1, with around 70-fold selectivity for OX1 over OX2 receptors.
• (0)
• (0)

• S1553
• ABT-492
• ABT-492 is a new fluoroquinolone against 155 aerobic and 171 anaerobic pathogens.
• (0)
• (0)

• S1516
• Cidofovir(Vistide)
• Cidofovir(Vistide) is an injectable antiviral medication for the treatment of cytomegalovirus (CMV) retinitis. (IC50= 0.94 μM).
• (0)
• (0)

• S1501
• Mycophenolate mofetil (CellCept)
• Mycophenolate mofetil is a inhibitor of inosine monophosphate dehydrogenase and a immunosuppressant.
• (0)
• (0)

• S1466
• Calcitriol (Rocaltrol)
• Calcitriol is the hormonally active form of vitamin D.
• (0)
• (0)

• S1464
• Marbofloxacin
• Marbofloxacin is a potent antibiotic of the fluoroquinolone group.
• (0)
• (0)

• S1448
• Azalomycin-B
• Azalomycin-B(Elaiophylin) is a macrolide antibiotic produced by Streptomyces hygroscopicus.
• (0)
• (0)

• S1450
• Nanchangmycin
• Nanchangmycin structurally and biologically resembles dianemycin, which is used in poultry farming.
• (0)
• (0)

• S1408
• Linezolid (Zyvox)
• Linezolid (Zyvox) is a synthetic antibiotic used for the treatment of serious infections.
• (0)
• (0)

• S1373
• Daptomycin
• Daptomycin is a novel lipopeptide antibiotic.
• (0)
• (0)

• S1374
• Doripenem Hydrate
• Doripenem (doripenem monohydrate) is an ultra-broad spectrum injectable antibiotic.
• (0)
• (0)

• S1312
• Streptozotocin (Zanosar)
• Streptozotocin(Streptozocin, Zanosar, STZ) is a naturally occurring chemical used in cancer chemotherapy and Type 1 diabetes treatment.
• (0)
• (0)

• S1290
• Celastrol
• Celastrol, a plant-derived triterpene, has anti-inflammatory and immunosuppressive activity.
• (0)
• (0)

• S1259
• Ramelteon (TAK-375)
• Ramelteon is a melatonin receptor agonist with both high affinity for melatonin MT1 (IC50 =28.5 ± 8.55 pM)and MT2 (20.1 ± 9.25 pM)receptors and selectivity over the MT3 receptor
• (0)
• (0)

• S1255
• Nepafenac
• Nepafenac is a non-steroidal anti-inflammatory agent.
• (0)
• (0)

• S1247
• Leflunomide
• Immunosuppressant agent. Its active metabolite is A77 1726 (RS-61980).
• (0)
• (0)

• S1211
• Imiquimod
• Imiquimod(Aldara) is a novel synthetic agent with immune response modifying activity.
• (0)
• (0)

• S1212
• Bendamustine HCL
• Bendamustine inhibits SU-DHL-1 cell proliferation with IC50 at 50 μm.
• (0)
• (0)

• S1222
• Dexrazoxane Hydrochloride
• A cardioprotective agent
• (0)
• (0)

• S1201
• Dimesna
• Dimesna (BNP7787, Tavocept, BioNumerik) is a uroprotective agent used in combination with cancer chemotherapeutic compounds to decrease urotoxicity.
• (0)
• (0)

• S1189
• Aprepitant (MK-0869)
• Substance P antagonists (SPA).
• (0)
• (0)

• P1082
• pp60 c-src (521-533)(phosphorylated)
• SRC kinase inhibitor
• (0)
• (0)

• P1081
• JIP-1(153-163)
• JNK and p38 MAPK inhibitor
• (0)
• (0)

• P1080
• Bax inhibitor peptide,negative control
• Bax inhibitor peptide,negative control is a negative control peptide for the Bax inhibitor peptides V5 and P5.
• (0)
• (0)

• P1077
• [Ala92]-p16 (84-103)
• [Ala92]-p16 (84-103) is a CDK inhibitor with IC50 of 1.5μM for cyclin-dependent kinase-4 (cdk4)/cyclin D1
• (0)
• (0)

• S1137
• Malotilate
• Malotilate is a liver protein metabolism improved compound.
• (0)
• (0)

• S1115
• Odanacatib (MK 0822)
• cathepsin K inhibitor with an IC50 of 0.2nM.
• (0)
• (0)

• S1097
• BTZ043 racemate
• BTZ043 racemate is a decaprenylphosphoryl-b-D-ribose 2’-epimerase inhibitor with MIC of 2.3 and 9.2 nM for M. tuberculosis H37Rv and Mycobacterium smegmatis, respectively.
• (0)
• (0)

• S1041
• STF-62247
• Targeting VHL-deficient RCC cells, in renal cell carcinoma (RCC) cells that have lost the von Hippel-Lindau (VHL) tumor suppressor activity (IC50 = 625 μM).
• (0)
• (0)

• S5004
• Pimecrolimus
• Inhibitor of inflammatory cytokine secretion
• (0)
• (0)

• S6002
• NXY-059 (Cerovive)
• NXY-059 (Cerovive) is the disulfonyl derivative of the neuroprotective spin trap phenylbutynitrone or "PBN".
• (0)
• (0)